
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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Ac-YVAD-AOM
CAS:Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.Formula:C33H42N4O10Purity:98%Color and Shape:SolidMolecular weight:654.71β-Anhydroicaritin
CAS:β-Anhydroicaritin is a natural product extracted from Boswellia serrata with anti-osteoporosis, estrogen regulation and anti-tumour properties.Formula:C21H20O6Purity:96.95%Color and Shape:SolidMolecular weight:368.38PD-166793
CAS:PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.Formula:C17H18BrNO4SPurity:100%Color and Shape:SolidMolecular weight:412.3Ref: TM-T20563
2mg57.00€5mg87.00€10mg137.00€25mg274.00€50mg439.00€100mg658.00€500mg1,359.00€1mL*10mM (DMSO)97.00€3-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-, methanesulfonate (1:1)
CAS:Formula:C33H49N3O7S2Purity:96%Color and Shape:SolidMolecular weight:663.8881JNJ0966
CAS:JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).Formula:C16H16N4O2S2Purity:99.46% - 99.48%Color and Shape:SolidMolecular weight:360.45Ref: TM-T4783
1mg39.00€5mg64.00€10mg96.00€25mg183.00€50mg329.00€100mg475.00€200mg655.00€1mL*10mM (DMSO)50.00€Azt-pmap
CAS:AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].Formula:C20H25N6O8PPurity:98%Color and Shape:SolidMolecular weight:508.42Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Formula:C25H26N7O8PPurity:98.95%Color and Shape:SolidMolecular weight:583.49Ref: TM-T3523
1mg59.00€5mg120.00€10mg170.00€25mg283.00€50mg432.00€100mg622.00€200mg873.00€1mL*10mM (DMSO)156.00€Phepropeptin D
CAS:Phepropeptin D is a secondary metabolite produced by microorganisms and acts as a proteasome (proteasome) inhibitor, with an IC50 of 7.8 μg/mL.Formula:C41H58N6O6Color and Shape:SolidMolecular weight:730.94Pseudostellarin G
CAS:Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.Formula:C42H56N8O9Color and Shape:SolidMolecular weight:816.94Benzenemethanesulfonyl fluoride
CAS:Formula:C7H7FO2SPurity:99%Color and Shape:SolidMolecular weight:174.1927Ref: IN-DA00I6AP
1g25.00€5g39.00€10g55.00€1kgTo inquire25g93.00€2kgTo inquire50g137.00€5kgTo inquire100g181.00€250g572.00€500gTo inquireAc-FLTD-CMK
CAS:Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.Formula:C26H37ClN4O8Purity:95.17%Color and Shape:SolidMolecular weight:569.05Marimastat
CAS:Marimastat (BB2516) (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C15H29N3O5Purity:97.46% - 98.11%Color and Shape:SolidMolecular weight:331.41Cytochalasin H
CAS:Cytochalasin H ((16-Benzyl-5,12-dihydroxy-5,7,14-trimethyl-13-methylidene-18-oxo-17-azatricyclo[9.7.0.01,15]octadeca-3,9-dien-2-yl) acetate) is a potentFormula:C30H39NO5Purity:98.04%Color and Shape:SolidMolecular weight:493.63Ref: TM-T21513
1mg97.00€2mg142.00€5mg226.00€10mg340.00€25mg553.00€50mg735.00€100mg1,008.00€200mg1,359.00€1mL*10mM (DMSO)415.00€N-Phenylthiourea
CAS:N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.Formula:C7H8N2SPurity:99.71%Color and Shape:SolidMolecular weight:152.22MMP2-IN-2
CAS:MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.Formula:C13H8N4O4Purity:98.09%Color and Shape:SolidMolecular weight:284.23HIV-1 protease-IN-12
CAS:HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-Formula:C25H35N3O5SPurity:98%Color and Shape:SolidMolecular weight:489.63Ac-VRPR-AMC TFA
Ac-VRPR-AMC TFA serves as a fluorogenic substrate for metacaspases, enabling the assay of metacaspase activity.Formula:C38H53F6N11O11Color and Shape:SolidMolecular weight:953.88Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formula:C41H52N4O4SPurity:97.87%Color and Shape:SolidMolecular weight:696.94Ref: TM-TQ0297
1mg69.00€5mg149.00€10mg235.00€25mg470.00€50mg610.00€100mg793.00€200mg1,064.00€1mL*10mM (DMSO)221.00€MDL-28170
CAS:MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.Formula:C22H26N2O4Purity:98%Color and Shape:SolidMolecular weight:382.45Ref: TM-T2470
1mg35.00€2mg52.00€5mg74.00€10mg96.00€25mg135.00€50mg177.00€100mg299.00€1mL*10mM (DMSO)80.00€Deapioplatycodin D
CAS:Deapioplatycodin D and platycodin D can regulate the production and secretion of airway mucin and, explains the use of aqueous extract of APG as expectorants.Formula:C52H84O24Purity:99.11% - 99.64%Color and Shape:SolidMolecular weight:1093.21