
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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Dabigatran Etexilate Mesylate
CAS:Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.Formula:C34H41N7O5·CH4O3SPurity:99.91%Color and Shape:SolidMolecular weight:723.84Ref: TM-T5133
5mg42.00€10mg57.00€25mg74.00€50mg95.00€100mg111.00€200mg169.00€500mg240.00€1mL*10mM (DMSO)64.00€NM107
CAS:NM107, a ribonucleoside, inhibits HCV NS5B polymerase. It has broad antiviral properties with EC50 of 1.85 μM in wild-type cells.Formula:C10H15N3O5Purity:98%Color and Shape:White To Off-White PowderMolecular weight:257.24MRS1177
CAS:MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).Formula:C20H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:389.79Methyl rosmarinate
CAS:Methyl rosmarinate, from Rabdosia serra, inhibits tyrosinase (IC50: 0.28 mM), α-glucosidase, MMP-1, and has antioxidant, antifungal properties.Formula:C19H18O8Purity:97.52% - 99.62%Color and Shape:SolidMolecular weight:374.34Ref: TM-TN1928
1mg74.00€5mg165.00€10mg259.00€25mg435.00€50mg630.00€100mg880.00€1mL*10mM (DMSO)173.00€GLS1 Inhibitor-4
CAS:GLS1 Inhibitor-4 (41e) has 11.86 nM IC50, strong binding, disrupts glutamine metabolism, induces apoptosis, and shows antitumor effects.Formula:C29H27F3N10O2S2Purity:98%Color and Shape:SolidMolecular weight:668.72Collagenase Type IV
Collagenase Type IV is an MMP-18 primarily degrades collagen type IV and VII and basement membranes (e.g., neural tissue, renal tissue) mild activity.Color and Shape:Odour SolidMirificin
CAS:Mirificin (BCP10902) is an active ingredient in Tongmai formula (TMF) which is a well-known Chinese medicinal preparation. Anti-oxidant.Formula:C26H28O13Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:548.49Ubenimex
CAS:Formula:C16H24N2O4Purity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:308.38Eltrombopag
CAS:Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the plateletFormula:C25H22N4O4Purity:99.27%Color and Shape:Orange To Red SolidMolecular weight:442.471,10-Phenanthroline Monohydrate [for Biochemical Research]
CAS:Formula:C12H8N2·H2OPurity:>99.0%(T)Color and Shape:White powder to crystalMolecular weight:198.23HIV-1 integrase inhibitor 8
CAS:HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].Formula:C21H24O2Purity:98.01%Color and Shape:SolidMolecular weight:308.41Monobenzone
CAS:Monobenzone (Benoquin) is a Depigmenting Agent.Formula:C13H12O2Purity:99.87%Color and Shape:Lustrous Leaflets From Water SolidMolecular weight:200.23Aclacinomycin A hydrochloride
CAS:Aclacinomycin A (Aclarubicin) hydrochloride is a fluorescent molecule and the first described non-peptidic inhibitor showing discrete specificity for the CTRL (Formula:C42H54ClNO15Purity:98%Color and Shape:SolidMolecular weight:848.33Ref: TM-T10238
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire200mgTo inquire1mL*10mM (DMSO)To inquireVCH-916 free acid(1200133-34-1 free base)
CAS:VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Formula:C26H37NO4SPurity:98.45%Color and Shape:SolidMolecular weight:459.64Ref: TM-TQ0122L
1mg74.00€2mg97.00€5mg140.00€10mg188.00€25mg339.00€50mg552.00€100mg792.00€1mL*10mM (DMSO)150.00€BI-1230
CAS:BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.Formula:C42H52N6O9SPurity:98%Color and Shape:SolidMolecular weight:816.96TGase2-IN-1
CAS:TGase2-IN-1 (Compound 22) is an orally effective TGase2 inhibitor with an IC50 of 1.12 µM. It inhibits TGase2 in human retinal microvascular endothelial cells with a strikingly lower IC50 of 0.07 µM. The oral bioavailability of TGase2-IN-1 is 74.6%. Additionally, it can suppress retinal vascular leakage in a mouse model of diabetes induced by Streptozotocin.Formula:C23H25N3O3Color and Shape:SolidMolecular weight:391.46Cathepsin Inhibitor 2
CAS:Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).Formula:C19H21F6N3OPurity:98%Color and Shape:SolidMolecular weight:421.38Temocapil
CAS:Temocapril is an inhibitor of tyrosine kinase.Formula:C23H28N2O5S2Purity:97.8%Color and Shape:White PowderMolecular weight:476.61IK-862
CAS:IK-862 is a selective TACE inhibitor with potential anti-inflammatory and anticancer activity for the study of neuritis.Formula:C25H27N3O4Purity:98.72% - 99.39%Color and Shape:SolidMolecular weight:433.5MK-0608
CAS:MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).Formula:C12H16N4O4Purity:98.48%Color and Shape:SolidMolecular weight:280.28Ref: TM-T16088
1mg81.00€2mg96.00€5mg170.00€10mg274.00€25mg525.00€50mg753.00€100mg1,035.00€1mL*10mM (DMSO)183.00€