
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
Show 4 more subcategories
Products of "Proteases/Proteasome"
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Excisanin A
CAS:ExcisaninA may be a potent inhibitor of AKT signaling pathway in tumor cells, it can inhibit invasion by suppressing MMP-2 and MMP-9 expression, it may be aFormula:C20H30O5Purity:98%Color and Shape:SolidMolecular weight:350.45S 3304
CAS:S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.Formula:C24H20N2O4S2Purity:98.09%Color and Shape:SolidMolecular weight:464.56Ref: TM-T16966
1mg58.00€5mg160.00€10mg259.00€25mg429.00€50mg605.00€100mg815.00€200mg1,093.00€1mL*10mM (DMSO)163.00€Reverse transcriptase-IN-1
CAS:Reverse transcriptase-IN-1 is a diarylbenzopyrimidine (DABP) analogue and a potent inhibitor of HIV-1 nonnucleoside reverse transcriptase with an IC50of 13.7Formula:C25H17N7O2Purity:99.14%Color and Shape:SolidMolecular weight:447.45Ref: TM-T12715
1mg64.00€5mg131.00€10mg183.00€25mg311.00€50mg449.00€100mg615.00€200mg833.00€1mL*10mM (DMSO)143.00€MMP-9-IN-1
CAS:MMP-9-IN-1 is an inhibitor of specific matrix metalloproteinase-9 (MMP-9).Formula:C16H17F2N3O3SPurity:99.21%Color and Shape:SolidMolecular weight:369.39Ref: TM-T8310
1mg96.00€2mg139.00€5mg227.00€10mg359.00€25mg607.00€50mg847.00€100mg1,169.00€1mL*10mM (DMSO)221.00€ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formula:C23H18ClF3N4O2S2Purity:98%Color and Shape:SolidMolecular weight:538.99Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formula:C22H30N6OSPurity:99.73%Color and Shape:SolidMolecular weight:426.58Ref: TM-T37522
1mgTo inquire5mg35.00€10mg52.00€25mg74.00€50mg97.00€100mg173.00€200mgTo inquire1mL*10mM (DMSO)50.00€Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Formula:C19H17NO7Purity:97.99%Color and Shape:SolidMolecular weight:371.34Tyrosinase-IN-36
Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.Color and Shape:Odour SolidDabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purity:97.63%Color and Shape:SolidMolecular weight:499.56Diprotin A
CAS:Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formula:C17H31N3O4Purity:99.29%Color and Shape:White PowderMolecular weight:341.45Ginkgolide C
CAS:Ginkgolide C (BN-52022), a natural product, can enhance the cardiac function of rats in the body.Formula:C20H24O11Purity:99.71% - 99.98%Color and Shape:White PowderMolecular weight:440.4Phepropeptin B
CAS:Phepropeptin B is a secondary metabolite derived from microorganisms, functioning as a proteasome (proteasome) inhibitor with an IC50 value of 11 μg/mL.Formula:C40H56N6O6Color and Shape:SolidMolecular weight:716.91Eltrombopag Olamine
CAS:Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietinFormula:C29H36N6O6Purity:99.59% - 99.89%Color and Shape:SolidMolecular weight:564.63Ref: TM-T6825
2mg43.00€5mg64.00€10mg90.00€25mg140.00€50mg177.00€100mg230.00€200mg340.00€500mg563.00€1mL*10mM (DMSO)90.00€MUN57694
CAS:MUN57694 is an inhibitor of 26S proteasome.Formula:C23H25N3O4Purity:99%Color and Shape:SolidMolecular weight:407.46Ref: TM-T9090
1mg40.00€5mg80.00€10mg116.00€25mg212.00€50mg316.00€100mg447.00€200mg627.00€1mL*10mM (DMSO)96.00€Obefazimod
CAS:Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).Formula:C16H10ClF3N2OPurity:99.86%Color and Shape:SolidMolecular weight:338.71Ref: TM-T8311
2mg39.00€5mg62.00€10mg87.00€25mg187.00€50mg301.00€100mg437.00€200mg617.00€1mL*10mM (DMSO)65.00€Trovirdine
CAS:Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.Formula:C13H13BrN4SPurity:98.12% - 98.50%Color and Shape:SolidMolecular weight:337.24HZ-1157
CAS:HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.Formula:C12H16N4OPurity:98.23%Color and Shape:SolidMolecular weight:232.28UPGL00004
CAS:UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Formula:C25H26N8O2S2Purity:97.44%Color and Shape:SolidMolecular weight:534.66Ginsenoside F4
CAS:Ginsenoside F4 induces apoptosis in JK cells by causing mitochondrial dysfunction and altering Bax and Bcl-2 levels.Formula:C42H70O12Purity:98%Color and Shape:SolidMolecular weight:767.01Feniralstat
CAS:Feniralstat (KVD-824) is a selective and potent kallikrein (kallikrein) inhibitor, useful in immune system diseases and cardiovascular disease research.Formula:C26H25F2N5O4Purity:99.52%Color and Shape:SolidMolecular weight:509.51