CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 4 more subcategories

Products of "Proteases/Proteasome"

Sort by

products per page.Found 857 products on this category.
  • Ac-VRPR-AMC

    CAS:
    Ac-VRPR-AMC is a fluorogenic substrate for metacaspase activity assays, facilitating the detection and measurement of metacaspase activity [1].
    Formula:C34H51N11O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:725.84

    Ref: TM-T80110

    5mg
    To inquire
    50mg
    To inquire
  • 2-PMPA

    CAS:
    2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).
    Formula:C6H11O7P
    Purity:98% - 99.50%
    Color and Shape:Solid
    Molecular weight:226.12

    Ref: TM-T3440

    5mg
    66.00€
    10mg
    93.00€
    25mg
    180.00€
    50mg
    259.00€
    100mg
    430.00€
  • Tyrosinase-IN-32


    Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.
    Formula:C15H19NO3
    Color and Shape:Solid
    Molecular weight:261.32

    Ref: TM-TN8160

    10mg
    To inquire
    50mg
    To inquire
  • ABT530

    CAS:
    ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.
    Formula:C57H65F5N10O8
    Purity:99.15% - 99.93%
    Color and Shape:Solid
    Molecular weight:1113.18

    Ref: TM-T5127

    10mg
    48.00€
    25mg
    88.00€
    50mg
    127.00€
    100mg
    188.00€
    1mL*10mM (DMSO)
    52.00€
  • MMP-3 Inhibitor

    CAS:
    MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.
    Formula:C27H46N10O9S
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:686.78

    Ref: TM-T37048

    1mg
    81.00€
    5mg
    208.00€
    10mg
    309.00€
    25mg
    525.00€
    50mg
    757.00€
    100mg
    1,035.00€
    500mg
    2,110.00€
    1mL*10mM (DMSO)
    221.00€
  • Isoangustone A

    CAS:
    Isoangustone A has antitumor activity, it can induce G1 cycle arrest in DU145 human prostate and 4T1 murine mammary cancer cells, it inhibits cell proliferation
    Formula:C25H26O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.47

    Ref: TM-TN4263

    1mg
    513.00€
  • MMP13-IN-3

    CAS:
    MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.
    Formula:C24H22N4O5
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:446.46

    Ref: TM-T16124

    1mg
    87.00€
    5mg
    216.00€
    10mg
    354.00€
    25mg
    620.00€
    50mg
    847.00€
    100mg
    1,169.00€
    1mL*10mM (DMSO)
    240.00€
  • N-α-Tosyl-L-lysine chloromethyl ketone hydrochloride

    CAS:
    N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride inhibits trypsin-like proteases and IFN-γ activities.
    Formula:C14H22Cl2N2O3S
    Purity:97.44%
    Color and Shape:Powder
    Molecular weight:369.31

    Ref: TM-T16169

    5mg
    52.00€
    10mg
    81.00€
    25mg
    123.00€
    50mg
    177.00€
    1mL*10mM (DMSO)
    74.00€
  • TNF Protease Inhibitor 2

    CAS:
    TAPI-2 is a broad-spectrum inhibitor of MMP (IC50: 20 μM), tumour necrosis factorα-converting enzyme (TACE) and a disintegrin and metalloproteinase (ADAM).
    Formula:C19H37N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.53

    Ref: TM-TQ0129

    5mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • MG-132

    CAS:
    Formula:C26H41N3O5
    Purity:>95.0%(qNMR)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:475.63

    Ref: 3B-M3244

    10mg
    123.00€
  • Z-Leu-Leu-Tyr-COCHO

    CAS:
    Z-Leu-Leu-Tyr-COCHO is a potent inhibitor of chymotrypsin-like activity, exhibiting a Ki value of 3.0 nM [1].
    Formula:C30H39N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.65

    Ref: TM-T80102

    5mg
    To inquire
    50mg
    To inquire
  • Emivirine

    CAS:
    Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.
    Formula:C17H22N2O3
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:302.37

    Ref: TM-T27260

    1mg
    35.00€
    5mg
    80.00€
    10mg
    116.00€
    25mg
    188.00€
    50mg
    To inquire
    1mL*10mM (DMSO)
    87.00€
  • Benzylsulfonyl Fluoride [for Biochemical Research]

    CAS:
    Formula:C7H7FO2S
    Purity:>98.0%(GC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:174.19

    Ref: 3B-B3473

    5g
    51.00€
    25g
    131.00€
  • BI 224436

    CAS:
    BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.
    Formula:C27H26N2O4
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T14559

    1mg
    4,874.00€
    5mg
    9,377.00€
  • HIV-1 protease-IN-9

    CAS:
    HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a
    Formula:C37H41N7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:679.83

    Ref: TM-T79295

    5mg
    1,301.00€
    50mg
    2,642.00€
    100mg
    3,515.00€
  • CDK9-IN-30

    CAS:
    CDK9-IN-30 is one of the Tat peptide derivatives and inhibits HIV-1 long terminal repeat-activated transcription.
    Formula:C16H20FNO3
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:293.33

    Ref: TM-T9632

    1mg
    56.00€
    5mg
    119.00€
    10mg
    187.00€
    25mg
    316.00€
    50mg
    472.00€
    100mg
    658.00€
    500mg
    1,378.00€
    1mL*10mM (DMSO)
    114.00€
  • GLPG2451

    CAS:
    GLPG2451 potentiates F508del CFTR at low temp (EC50: 11.1 nM), aiding cystic fibrosis treatment.
    Formula:C16H16F3N3O5S
    Color and Shape:Solid
    Molecular weight:419.38

    Ref: TM-T13705

    5mg
    283.00€
    25mg
    938.00€
    50mg
    1,293.00€
    100mg
    1,768.00€
    1mL*10mM (DMSO)
    346.00€
  • Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]

    CAS:
    Formula:C10H13N2Na3O8·xH2O
    Purity:>98.0%(T)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:358.19 (as Anhydrous)

    Ref: 3B-T2599

    5g
    22.00€
    25g
    41.00€
  • Benzoic acid, 4-[(aminoiminomethyl)amino]-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate

    CAS:
    Formula:C21H25N5O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.5819

    Ref: IN-DA003SPE

    1g
    175.00€
    5g
    To inquire
    10mg
    25.00€
    50mg
    48.00€
    250mg
    100.00€
  • MMP-2 Inhibitor-4


    MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).
    Formula:C19H23N3O5S
    Molecular weight:405.468

    Ref: TM-T204609

    10mg
    To inquire
    50mg
    To inquire