
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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Sofosbuvir impurity H
Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.Formula:C29H33FN3O10PPurity:98%Color and Shape:SolidMolecular weight:633.56Licraside
CAS:Licraside is a tyrosinase inhibitor with an IC50 of 0.072 mM for monophenolase and can be used in studies about antibrowning and depigmenting agents.Formula:C26H30O13Purity:99.85%Color and Shape:SolidMolecular weight:550.51Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurity:98% - 99.55%Color and Shape:Off-White SolidMolecular weight:482.51Cilastatin
CAS:Cilastatin (MK0791): protects imipenem from renal breakdown; inhibits leukotriene D4 metabolism.Formula:C16H26N2O5SPurity:97.76% - 99.71%Color and Shape:SolidMolecular weight:358.45Ref: TM-T2583
5mg35.00€10mg44.00€25mg63.00€50mg88.00€100mg124.00€200mg188.00€500mg325.00€1mL*10mM (DMSO)55.00€Flovagatran
CAS:Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.Formula:C27H36BN3O7Purity:99.56%Color and Shape:SolidMolecular weight:525.4Ro24-7429
CAS:Ro24-7429: oral HIV-1 Tat antagonist, RUNX1 inhibitor with anti-HIV, antifibrotic, and anti-inflammatory properties.Formula:C14H13ClN4Purity:99.29% - 99.85%Color and Shape:SolidMolecular weight:272.73Ref: TM-T28578
1mg92.00€5mg187.00€10mg298.00€25mg507.00€50mg730.00€100mg1,026.00€500mg2,877.00€1mL*10mM (DMSO)215.00€Caspase-3 activator 3
Caspase-3 activator 3 (compound 2h) effectively induces apoptosis in HL-60 and K562 cells by substantially activating caspase-3, demonstrating antileukemicPurity:98%Color and Shape:Odour Solid3-Aminobenzene-1,2-diol
CAS:3-Aminobenzene-1,2-diol (compound C8) is an inhibitor of matrix metalloproteinases (MMP), with IC50 values of 20, 26, 16, and 16.3 μM against MMP-2, MMP-8, MMP-9, and MMP-14, respectively.Formula:C6H7NO2Color and Shape:SolidMolecular weight:125.132-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purity:≥95%Color and Shape:SolidMolecular weight:208.21HIV-1 protease-IN-7
CAS:HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].Formula:C68H104N10O12SPurity:98%Color and Shape:SolidMolecular weight:1285.68Aderamastat
CAS:Aderamastat (FP-025) is an orally active matrix metalloproteinase 12 (MMP-12) inhibitor indicated for the study of allergic asthma, COPD and pulmonary fibrosis.Formula:C21H18N2O4SPurity:99.35%Color and Shape:SolidMolecular weight:394.44PF 00356231
CAS:PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).Formula:C25H20N2O3SPurity:99.35%Color and Shape:SolidMolecular weight:428.5R-1479
CAS:R-1479 (4'-Azidocytidine) is an RdRp inhibitor with an IC50 value of 1.28 μM for HCV RNA replication in the HCV subgenomic replicon system.Formula:C9H12N6O5Purity:99.68% - 99.95%Color and Shape:SolidMolecular weight:284.23Ref: TM-TQ0162
1mg135.00€2mg187.00€5mg329.00€10mg472.00€25mg753.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)363.00€Trypsin Inhibitor, soybean
CAS:Trypsin Inhibitor, soybean is a trypsin inhibitor extracted from leguminous plants.Color and Shape:SolidPhepropeptin C
CAS:Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.Formula:C38H60N6O6Color and Shape:SolidMolecular weight:696.92Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Formula:C13H17NO8Purity:99.52%Color and Shape:SolidMolecular weight:315.28Isoderrone
CAS:Isoderrone inhibits α-glucosidase and PTP1B; IC50 = 22.7 uM, potential type 2 diabetes drug.Formula:C20H16O5Purity:98%Color and Shape:SolidMolecular weight:336.34Tenofovir alafenamide hemifumarate
CAS:Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.Formula:C21H29N6O5PC4H4O4Purity:99.33% - 99.96%Color and Shape:SolidMolecular weight:534.51Glucosamine
CAS:Glucosamine (Chitosamine) is an amino sugar and a prominent precursor in the biochemical synthesis of glycosylated proteins and lipids.Formula:C6H13NO5Purity:99.80% - 99.80%Color and Shape:CoaMolecular weight:179.17S-Methylglutathione
CAS:S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.Formula:C11H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:321.35