
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
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Products of "Proteases/Proteasome"
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lavendustin B
CAS:Lavendustin B inhibits Tyrosine Kinase and HIV-1 integrase-LEDGF/p75 interaction.Formula:C21H19NO5Purity:95.72%Color and Shape:Off-White SolidMolecular weight:365.38Ref: TM-T4182
1mg62.00€2mg87.00€5mg119.00€10mg188.00€25mg425.00€50mg625.00€100mg892.00€1mL*10mM (DMSO)131.00€AMD 3465
CAS:AMD 3465 (GENZ-644494) blocks CXCR4, hinders X4 HIV replication (IC50: 1-10 nM), ineffective against R5 viruses, IC50: 0.75 nM (12G5 mAb), 18 nM (CXCL12AF647).Formula:C24H38N6Purity:98%Color and Shape:SolidMolecular weight:410.60ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Formula:C17H20N2O5SPurity:98.24%Color and Shape:SolidMolecular weight:364.426-Hydroxykaempferol
CAS:6-Hydroxykaempferol, a competitive tyrosinase inhibitor, a flavonoid, and a natural product, has higher activity than L-DOPA and high antioxidant activity.Formula:C15H10O7Purity:98%Color and Shape:SolidMolecular weight:302.24NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formula:C44H44N6O8Purity:98%Color and Shape:SolidMolecular weight:784.86Bivalirudin
CAS:Bivalirudin (BG-8967) is a reversible inhibitor of α- and ζ-thrombin (Kis = 2.56 and 1.84 nM, respectively), enzymes that exhibit high fibrinogen-clottingFormula:C98H138N24O33Purity:100.00% - 98.8%Color and Shape:White To Off-White PowderMolecular weight:2180.29Cynaropicrin
CAS:Cynaropicrin is a sesquiterpene lactone found in artichoke with anti-hepatitis C and trypanosome activity and inhibits NF-κB activation.Formula:C19H22O6Purity:96.15%Color and Shape:SolidMolecular weight:346.37Didanosine
CAS:Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).Formula:C10H12N4O3Purity:99.64%Color and Shape:White Crystalline PowderMolecular weight:236.23M867
CAS:M867 is a selective, reversible caspase-3 inhibitor, possessing an IC50 of 1.4 nM and a Ki value of 0.7 nM, demonstrating anti-apoptotic activity [1].Formula:C27H43N7O6Purity:98%Color and Shape:SolidMolecular weight:561.67Proteasome-IN-1
CAS:Proteasome-IN-1 is an inhibitor of proteasome.Formula:C42H35N5O3Purity:98%Color and Shape:SolidMolecular weight:657.76MG-115
CAS:MG-115 inhibits 20S (21 nM Ki) and 26S (35 nM Ki) proteasomes, targets chymotrypsin-like activity & induces p53 apoptosis.Formula:C25H39N3O5Purity:97.12%Color and Shape:White PowderMolecular weight:461.592'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purity:99.93%Color and Shape:SolidMolecular weight:383.83Sofosbuvir impurity A
CAS:Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.Formula:C22H29FN3O9PPurity:98%Color and Shape:SolidMolecular weight:529.45Benzenesulfonyl fluoride, 4-(2-aminoethyl)-, hydrochloride (1:1)
CAS:Formula:C8H11ClFNO2SPurity:98%Color and Shape:SolidMolecular weight:239.6948CA-074 methyl ester
CAS:CA-074 methyl ester (Cathepsin B Inhibitor IV) is a specific inhibitor of Cathepsin B with neuroprotective, anti-cancer, and anti-inflammatory effects.Formula:C19H31N3O6Purity:97.26% - 99.58%Color and Shape:SolidMolecular weight:397.47Ref: TM-T3420
1mg59.00€2mg79.00€5mg115.00€10mg178.00€25mg360.00€50mg532.00€100mg743.00€200mg1,026.00€1mL*10mM (DMSO)96.00€Sivelestat Sodium Tetrahydrate
CAS:Formula:C20H21N2NaO7S·4H2OPurity:>95.0%(T)(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:528.50Z-Ala-Ala-Asp-CMK
CAS:Z-Ala-Ala-Asp-chloromethylketone (Z-AAD-CMK) is a selective inhibitor of granzyme B [1].Formula:C19H24ClN3O7Purity:98%Color and Shape:SolidMolecular weight:441.86HIV-1 inhibitor-54
CAS:HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.Formula:C27H30N6O4SPurity:97.61% - 98.61%Color and Shape:SoildMolecular weight:534.63Menadione
CAS:Menadione (Vitamin K3) is a synthetic naphthoquinone, inactive but converts to active Vitamin K2 in vivo.Formula:C11H8O2Purity:99.08% - 99.41%Color and Shape:Bright Yellow Crystals SolidMolecular weight:172.18