Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Products of "Opioid Receptor"
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CP 866087
CAS:CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H30N2O3SPurity:99.28% - 99.52%Color and Shape:SolidMolecular weight:426.57Norbinaltorphimine dihydrochloride
CAS:Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.Formula:C40H45Cl2N3O6Purity:99%Color and Shape:SolidMolecular weight:734.71Endomorphin 1
CAS:Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).Formula:C34H38N6O5Purity:95.92%Color and Shape:Solid (Solid Powder )Molecular weight:610.7JNJ-20788560
CAS:JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).Formula:C25H28N2O2Purity:98.00%Color and Shape:SolidMolecular weight:388.5BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Formula:C30H31BrO4Purity:98.76%Color and Shape:SolidMolecular weight:535.47Fluorphine
CAS:Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.Formula:C20H22FN3OColor and Shape:SolidMolecular weight:339.41Naltrindole 5′-isothiocyanate
CAS:Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.Formula:C27H25N3O3SColor and Shape:SolidMolecular weight:471.571SCH-486757
CAS:SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.Formula:C24H23Cl2N3OPurity:100% - 99.53%Color and Shape:SolidMolecular weight:440.37ORL1 antagonist 1
CAS:ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).Formula:C20H22ClN5Purity:97.87%Color and Shape:SolidMolecular weight:367.88Ref: TM-T12320
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg475.00€100mg638.00€200mg845.00€1mL*10mM (DMSO)163.00€GSK1521498 free base
CAS:GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor.Formula:C24H20F2N4Purity:98%Color and Shape:SolidMolecular weight:402.44Isotodesnitazene
CAS:Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 values of 34.8 nM and 142 nM for MOR-βarr2 and MOR-mini-Gi, respectively. Isotodesnitazene can be utilized for research in opioid drugs.Formula:C23H31N3OColor and Shape:SolidMolecular weight:365.51BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formula:C18H25Cl3N2OPurity:99.04%Color and Shape:SolidMolecular weight:391.76Asimadoline hydrochloride
CAS:Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.Formula:C27H31ClN2O2Purity:98.94% - 99.32%Color and Shape:SolidMolecular weight:451.01Ref: TM-T4691
1mg35.00€5mg73.00€10mg111.00€25mg227.00€50mg338.00€100mg500.00€500mg1,074.00€1mL*10mM (DMSO)81.00€[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.Formula:C65H107N21O15Purity:99.05%Color and Shape:SoildMolecular weight:1422.7Sec-O-Glucosylhamaudol
CAS:Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.Formula:C21H26O10Purity:99.79%Color and Shape:SolidMolecular weight:438.43KOR agonist 4
KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.Formula:C21H25N3Color and Shape:SolidMolecular weight:319.44Bevenopran
CAS:Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.Formula:C20H26N4O4Purity:98.14% - 98.76%Color and Shape:SolidMolecular weight:386.44Ref: TM-T14551
1mg65.00€5mg137.00€10mg197.00€25mg316.00€50mg430.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)150.00€Alvimopan
CAS:Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.Formula:C25H32N2O4Purity:99.47% - 99.78%Color and Shape:SolidMolecular weight:424.53Ref: TM-T1242
1mg49.00€2mg69.00€5mg88.00€10mg139.00€25mg255.00€50mg378.00€100mg560.00€500mg1,216.00€1mL*10mM (DMSO)88.00€Icalcaprant
CAS:Icalcaprant is a kappa-opioid receptor antagonist [1].Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48AH 7959
CAS:AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.Formula:C19H26Cl2N2OColor and Shape:SolidMolecular weight:369.33
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