
p53
Los inhibidores de p53 se dirigen a la proteína p53, un supresor tumoral que desempeña un papel crucial en la regulación del ciclo celular, la reparación del ADN y la apoptosis. Aunque p53 a menudo está mutado o inactivado en células cancerosas, su inhibición a veces es necesaria para proteger a las células sanas de la apoptosis durante ciertos tratamientos. Por otro lado, restaurar la función de p53 en los tumores puede conducir a la apoptosis de las células cancerosas. La investigación sobre inhibidores de p53 es compleja y significativa tanto para comprender los mecanismos del cáncer como para desarrollar nuevas terapias. En CymitQuimica, ofrecemos una selección de inhibidores y moduladores de p53 de alta calidad para apoyar su investigación en biología del cáncer, apoptosis y desarrollo terapéutico.
Productos de "p53"
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BIX-01294
CAS:BIX-01294 is an G9a Histone Methyltransferase inhibitor(IC50 : 1.9 μM).Fórmula:C28H38N6O2Pureza:99.31% - 99.64%Forma y color:SolidPeso molecular:490.64Ref: TM-T7697
1mg40,00€2mg51,00€5mg85,00€10mg117,00€25mg207,00€50mg350,00€100mg518,00€200mg740,00€1mL*10mM (DMSO)131,00€Anti-p53 Antibody (9G129)
Anti-p53 Antibody (9G129) is a Rabbit antibody targeting p53. Anti-p53 Antibody (9G129) can be used in IHC-P,ICC/IF.Forma y color:Odour LiquidHLA-A*02:01&B2M&P53 R175H (HMTEVVRHC) Tetramer Protein, Human, MHC (His & Avi), PE-Labeled
p53 is a tumor suppressor protein.Forma y color:Odour Lyophilized PowderSCH529074
CAS:SCH529074 is a selective activator of p53 (Ki = 1 μM) and can be used in studies about non-small-cell lung carcinoma.Fórmula:C31H36Cl2N6Pureza:98.71%Forma y color:SolidPeso molecular:563.56Ref: TM-T37042
1mg35,00€2mg46,00€5mg64,00€10mg104,00€25mg220,00€50mg328,00€100mg469,00€1mL*10mM (DMSO)75,00€Schisandrol B
CAS:Schisandrol B fights neuroinflammation, liver/renal damage, and reduces cell growth via multiple signaling pathways.Fórmula:C23H28O7Pureza:99.14% - 99.32%Forma y color:SolidPeso molecular:416.46Ref: TM-T6S1917
5mg71,00€10mg96,00€25mg202,00€50mg303,00€100mg452,00€500mg1.035,00€1mL*10mM (DMSO)79,00€CTX1
CAS:CTX1 is a small molecule activator of p53.Fórmula:C14H10N4Pureza:98%Forma y color:SolidPeso molecular:234.26PDK4-IN-1 hydrochloride
CAS:PDK4-IN-1 hydrochloride is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4, IC50 value = 84 nM).Fórmula:C22H20ClN3O2Pureza:99.54%Forma y color:SolidPeso molecular:393.87Ref: TM-T12412L
1mg127,00€5mg300,00€10mg457,00€25mg750,00€50mg1.026,00€100mg1.406,00€500mg2.822,00€1mL*10mM (DMSO)329,00€Etoposide
CAS:Etoposide (VP-16-213) is a topoisomerase II inhibitor that inhibits DNA synthesis by forming a complex with topoisomerase II and DNA (IC50=60.3 μM).Fórmula:C29H32O13Pureza:99.19% - 99.94%Forma y color:Crystals From Methanol SolidPeso molecular:588.56Anti-p53 Antibody (9G324)
Anti-p53 Antibody (9G324) is an antibody targeting p53. Anti-p53 Antibody (9G324) can be used in ELISA, IF.Forma y color:Odour LiquidAmifostine thiol dihydrochloride
CAS:Amifostine (WR 1065) activates p53 via JNK and shields tissues from cancer drug toxicity.Fórmula:C5H16Cl2N2SPureza:100%Forma y color:SolidPeso molecular:207.165BML-259
CAS:BML-259 inhibits CDK5/CDK2 (IC50: 64/98 nM) for cancer and neurodegeneration research.Fórmula:C14H16N2OSPureza:99.68%Forma y color:SolidPeso molecular:260.35Ref: TM-T36964
5mg50,00€10mg85,00€25mg169,00€50mg279,00€100mg487,00€500mg1.035,00€1mL*10mM (DMSO)52,00€CT-1
CAS:CT-1 is a DNA minor groove ligand and causes p53-dependent breast cancer cell apoptosis.Fórmula:C29H23F3N4OPureza:99.24%Forma y color:SolidPeso molecular:500.51LLY-507
CAS:LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyltransferase SMYD2.Fórmula:C36H42N6OPureza:99.56% - 99.93%Forma y color:SolidPeso molecular:574.76Ref: TM-T6879
1mg44,00€2mg55,00€5mg85,00€10mg138,00€25mg304,00€50mg552,00€100mg787,00€1mL*10mM (DMSO)110,00€HLA-A*02:01&B2M&P53 R175H (HMTEVVRHC) Monomer Protein, Human, MHC (His & Avi), Biotinylated
p53 is a tumor suppressor protein.Forma y color:Odour Lyophilized Powder(S)-10-Hydroxycamptothecin
CAS:(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma.Fórmula:C20H16N2O5Pureza:99.09% - 99.81%Forma y color:SolidPeso molecular:364.35HLA-A*02:01&B2M&P53 R175H (HMTEVVRHC) Monomer Protein, Human, MHC (His & Avi)
p53 is a tumor suppressor protein.Forma y color:Odour Lyophilized PowderLeptomycin B
CAS:Leptomycin B: potent CRM1 inhibitor, blocks protein nuclear export and cell cycle, antifungal, modifies cysteine.Fórmula:C33H48O6Pureza:99.04% - 99.71%Forma y color:White Crystalline SolidPeso molecular:540.73Ref: TM-T15735
1mg202,00€2mg341,00€5mg620,00€10mg882,00€25mg1.320,00€50mg1.776,00€100mg2.403,00€1mL*10mM (DMSO)283,00€SLMP53-1
CAS:SLMP53-1 is a p53 activator with anti-tumor activity, activates reprogramming of glucose metabolism, and interferes with angiogenesis and migrationFórmula:C20H18N2O2Pureza:99.64%Forma y color:SolidPeso molecular:318.37Ref: TM-T60839
1mg126,00€5mg298,00€10mg487,00€25mg938,00€50mg1.568,00€100mg2.517,00€1mL*10mM (DMSO)35,00€NSC 66811
CAS:NSC 66811 inhibits MDM2-p53 interaction with 120 nM affinity, activating p53 in cancer cells.Fórmula:C23H20N2OPureza:96.94%Forma y color:SolidPeso molecular:340.42NSC 146109 hydrochloride
CAS:NSC 146109 hydrochloride is an activator of p53 targeting MDMX. NSC 146109 hydrochloride can be used for studies on breast cancer.Fórmula:C17H17ClN2SPureza:97.03%Forma y color:SolidPeso molecular:316.85