Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Azasetron hydrochloride
CAS:Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.Fórmula:C17H20ClN3O3·HClPureza:99.50%Forma y color:SolidPeso molecular:386.27Trimipramine maleate
CAS:Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Fórmula:C24H30N2O4Pureza:99.47%Forma y color:SolidPeso molecular:410.51Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.45% - 99.89%Forma y color:SolidPeso molecular:477.57Flumexadol
CAS:Flumexadol is a selective 5-HT2C receptor agonist with an affinity (Ki) of 25 nM for the (+)-enantiomer and exhibits 40-fold selectivity over the 5-HT2A receptor. It is an orally active, non-narcotic analgesic.Fórmula:C11H12F3NOPureza:98%Forma y color:SolidPeso molecular:231.21DREADD agonist 21
CAS:DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).Fórmula:C17H18N4Pureza:99.88%Forma y color:SolidPeso molecular:278.35Ref: TM-T11095L
2mg34,00€5mg58,00€10mg85,00€25mg140,00€50mg221,00€100mg329,00€200mg472,00€1mL*10mM (DMSO)52,00€Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Forma y color:White PowderPeso molecular:614.02Itasetron
CAS:Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.Fórmula:C16H20N4O2Pureza:100% - 99.63%Forma y color:SolidPeso molecular:300.364-Chloro-L-phenylalanine
CAS:4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases (TPH1 and TPH2).Fórmula:C9H10ClNO2Pureza:99.76% - 99.96%Forma y color:SolidPeso molecular:199.63Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Fórmula:C22H26N2O4Pureza:98% - 99.9%Forma y color:SolidPeso molecular:382.45Donitriptan
CAS:Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。Fórmula:C23H25N5O2Pureza:98.34%Forma y color:SolidPeso molecular:403.485-MeO-pyr-T
CAS:5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.Fórmula:C15H20N2OForma y color:SolidPeso molecular:244.33PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Fórmula:C21H29Cl2N3O4SPureza:98.50%Forma y color:SolidPeso molecular:490.44Naftidrofuryl oxalate
CAS:Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.Fórmula:C26H35NO7Pureza:97.12% - 98.38%Forma y color:SolidPeso molecular:473.567-Desmethyl-3-hydroxyagomelatine
CAS:7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Fórmula:C14H15NO3Pureza:98%Forma y color:SolidPeso molecular:245.27Etoperidone
CAS:Etoperidone is an antidepressant that acts as an orally active reuptake inhibitor for serotonin (serotonin) and noradrenaline (nor-adrenaline). It demonstrates specific binding affinities (Kd) for several receptors: 36 nM at the 5-HT2 receptor, 38 nM at the α1-adrenergic receptor (α1-adrenergic receptor), 85 nM at the 5-HT1A receptor, and 570 nM at the α2-adrenergic receptor (α2-adrenergic receptor).Fórmula:C19H28ClN5OForma y color:SolidPeso molecular:377.91Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Fórmula:C10H11ClF3N3Pureza:98.34%Forma y color:SolidPeso molecular:265.66Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Fórmula:C21H26ClN3OSPureza:99.3% - 99.72%Forma y color:SolidPeso molecular:403.97Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Forma y color:SolidPeso molecular:328.38Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Fórmula:C20H20NO4Pureza:97.18% - 99.06%Forma y color:SolidPeso molecular:338.38Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Fórmula:C19H21NPureza:99.05% - 99.23%Forma y color:SolidPeso molecular:263.38YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Fórmula:C14H17N3OPureza:98%Forma y color:SolidPeso molecular:243.38-OH-Dpat
CAS:8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Fórmula:C16H25NOPureza:98%Forma y color:SolidPeso molecular:247.38Ethylpropyltryptamine
CAS:Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Fórmula:C15H22N2Forma y color:SolidPeso molecular:230.35Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Fórmula:C24H32ClNO6Pureza:99.73%Forma y color:Colorless LiquidPeso molecular:465.97Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFórmula:C20H24N2O6SPureza:100%Forma y color:White PowderPeso molecular:420.48Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOForma y color:SolidPeso molecular:301.47NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H25N3O2SPureza:98%Forma y color:SolidPeso molecular:431.55AAZ-A 154 benzoate
CAS:AAZ-A 154 benzoate is a selective, competitive, and non-hallucinogenic 5-HT2AR antagonist. This compound facilitates neuronal growth in rodents and produces lasting beneficial behavioral effects.Fórmula:C21H26N2O3Forma y color:SolidPeso molecular:354.44Nardosinonediol
CAS:Nardosinonediol is a natural compound derived from Nardostachys jatamansi that acts as a SERT inhibitor, regulating serotonin levels and antidepressant.Fórmula:C15H24O3Pureza:98%Forma y color:SolidPeso molecular:252.35Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Fórmula:C19H19NSPureza:97.50%Forma y color:SolidPeso molecular:293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€SB-269970 hydrochloride
CAS:SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFórmula:C18H28N2O3S·HClPureza:98.45%Forma y color:SolidPeso molecular:388.95Ogerin
CAS:Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Fórmula:C17H17N5OPureza:99.50% - 99.75%Forma y color:SolidPeso molecular:307.35Ref: TM-T16378
1mg35,00€2mg52,00€5mg74,00€10mg115,00€25mg227,00€50mg380,00€100mg567,00€1mL*10mM (DMSO)86,00€Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.83%Forma y color:SolidPeso molecular:575.61Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Fórmula:C21H24N2Pureza:99.76%Forma y color:SolidPeso molecular:304.43PF-03382792
CAS:PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Fórmula:C23H32FN3O4Pureza:98.09%Forma y color:SolidPeso molecular:433.52NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Fórmula:C25H26ClN3O2SPureza:99.8%Forma y color:SoildPeso molecular:468.01Ref: TM-T12262L1
1mg52,00€5mg114,00€10mg172,00€25mg284,00€50mg411,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)138,00€Flesinoxan
CAS:Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Fórmula:C22H26FN3O4Forma y color:SolidPeso molecular:415.46Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Fórmula:C22H23N3O2Pureza:98.06% - 99%Forma y color:SolidPeso molecular:361.44VA012
CAS:VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. It has been shown to reduce food intake and prevent weight gain during subchronic administration without causing central nervous system-related discomfort. VA012 is applicable in obesity research.Fórmula:C21H19N3Forma y color:SolidPeso molecular:313.40Dapoxetine hydrochloride
CAS:Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.Fórmula:C21H23NO·HClPureza:99.5% - 99.70%Forma y color:White To Off-White Crystalline SolidPeso molecular:341.87Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFórmula:C20H24ClNPureza:97% - 99.94%Forma y color:Crystals White To Off-White PowderPeso molecular:313.865-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Fórmula:C16H21ClN4O3Pureza:98%Forma y color:SolidPeso molecular:352.82Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Fórmula:C23H24ClN3O2Pureza:99%Forma y color:SolidPeso molecular:409.91NPS ALX Compound 4a dihydrochloride
CAS:NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H27Cl2N3O2SPureza:98%Forma y color:SolidPeso molecular:504.47Facinicline hydrochloride
CAS:Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM).Fórmula:C15H19ClN4OPureza:99.72%Forma y color:SolidPeso molecular:306.79BIMU 8
CAS:BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Fórmula:C19H27ClN4O2Pureza:99.36%Forma y color:SolidPeso molecular:378.9Ref: TM-T21946
1mg89,00€5mg172,00€10mg249,00€25mg416,00€50mg615,00€100mg873,00€500mg1.768,00€1mL*10mM (DMSO)185,00€Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.Fórmula:C21H25ClN2O4SPureza:99.57%Forma y color:SolidPeso molecular:436.95BF-1
CAS:BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.Fórmula:C22H25NO2SPureza:100% - 99.25%Forma y color:SolidPeso molecular:367.50Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Fórmula:C18H22N2S·HBrPureza:100% - 99.89%Forma y color:SolidPeso molecular:379.36BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Fórmula:C14H18N2OPureza:98.07%Forma y color:SolidPeso molecular:230.31Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Fórmula:C21H26ClNPureza:99.99%Forma y color:Crystalline SolidPeso molecular:327.9Ref: TM-T4274
10mg47,00€25mg67,00€50mg87,00€100mg116,00€200mg170,00€500mg279,00€1mL*10mM (DMSO)50,00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Fórmula:C20H23Cl2F2N3O2Pureza:99.59%Forma y color:SolidPeso molecular:446.32Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Fórmula:C21H25NO4Pureza:100% - 99.8%Forma y color:Off-White SolidPeso molecular:355.43Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Fórmula:C24H27FN2O4Pureza:99.42%Forma y color:SolidPeso molecular:426.48EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Fórmula:C15H22N2OPureza:98.33% - 98.46%Forma y color:SolidPeso molecular:246.35Ref: TM-T11183
1mg92,00€2mg125,00€5mg170,00€10mg213,00€25mg474,00€50mg688,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)170,00€Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Fórmula:C17H26N4OPureza:98%Forma y color:SolidPeso molecular:302.41Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFórmula:C21H21ClN4OS·HCl·H2OPureza:98% - 99.83%Forma y color:Off-White PowderPeso molecular:467.12Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Fórmula:C28H36N4O2S·HClPureza:99.51%Forma y color:SolidPeso molecular:529.14(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Fórmula:C15H23NO2SPureza:99.81%Forma y color:SoildPeso molecular:281.41Ref: TM-T60027
1mg77,00€5mg155,00€10mg220,00€25mg338,00€50mg472,00€100mg632,00€200mg853,00€1mL*10mM (DMSO)163,00€Donitriptan hydrochloride
CAS:Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectivelyFórmula:C23H26ClN5O2Pureza:99.8% - 99.8%Forma y color:SolidPeso molecular:439.94Ref: TM-T21666
2mg40,00€5mg49,00€10mg64,00€25mg135,00€50mg240,00€100mg339,00€200mg439,00€500mgA consultarSumatriptan succinate
CAS:Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Fórmula:C18H27N3O6SPureza:97.53% - 99.51%Forma y color:White PowderPeso molecular:413.49Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Fórmula:C20H20ClNO4Pureza:99.79%Forma y color:SolidPeso molecular:373.8rac Desmethyl Citalopram Hydrochloride
CAS:rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.Fórmula:C19H20ClFN2OPureza:96.14%Forma y color:SolidPeso molecular:346.83Tegaserod
CAS:Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Fórmula:C16H23N5OPureza:99.89%Forma y color:SolidPeso molecular:301.39Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.5%Forma y color:SolidPeso molecular:492.68PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Pureza:98%Forma y color:Odour SolidAlprenolol
CAS:Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1AFórmula:C15H23NO2Pureza:99.73% - 99.78%Forma y color:SolidPeso molecular:249.35Mebhydrolin napadisylate
CAS:Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.77%Forma y color:White Or Almost White CrystallinePeso molecular:420.52Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Fórmula:C15H20ClN3O2·HClPureza:98.32%Forma y color:SolidPeso molecular:346.26Ref: TM-T5336
1mg46,00€5mg87,00€10mg144,00€25mg283,00€50mg454,00€100mg655,00€200mg930,00€1mL*10mM (DMSO)97,00€Protriptyline hydrochloride
CAS:Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.Fórmula:C19H21N·HClPureza:98.54% - 99.98%Forma y color:SolidPeso molecular:299.84Sulamserod
CAS:Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular relatedFórmula:C19H28ClN3O5SPureza:98.76%Forma y color:SolidPeso molecular:445.965-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Fórmula:C22H29FN4O2Pureza:99.25%Forma y color:SolidPeso molecular:400.49Ref: TM-T12597
1mg678,00€5mg1.359,00€10mg1.833,00€25mg2.727,00€50mg3.676,00€100mg4.969,00€1mL*10mM (DMSO)1.605,00€Lumateperone
CAS:Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Fórmula:C24H28FN3OPureza:99.77%Forma y color:SolidPeso molecular:393.5Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Fórmula:C22H20ClN3Pureza:99% - 99.66%Forma y color:SolidPeso molecular:361.87Masupirdine mesylate
CAS:Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's diseaseFórmula:C23H32BrN3O9S3Pureza:99.48%Forma y color:SolidPeso molecular:670.61Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Fórmula:C18H20N4Pureza:99.15%Forma y color:SolidPeso molecular:292.38SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFórmula:C15H14N4OPureza:99.61%Forma y color:SolidPeso molecular:266.3Ref: TM-T8357
1mg97,00€2mg150,00€5mg207,00€10mg311,00€25mg525,00€50mg757,00€100mg1.035,00€1mL*10mM (DMSO)216,00€AVN 322 free base
CAS:AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.Fórmula:C17H19N5O2SPureza:99.13%Forma y color:SolidPeso molecular:357.435-HT2A&5-HT2C agonist-1
CAS:5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.Fórmula:C14H20N2OPureza:98%Forma y color:SolidPeso molecular:232.325-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Fórmula:C24H26N4O2SPeso molecular:434.55Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Fórmula:C21H24BrN3O3SPureza:97.40% - 98.67%Forma y color:SolidPeso molecular:478.4Temanogrel
CAS:Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).Fórmula:C24H28N4O4Pureza:99.24%Forma y color:SolidPeso molecular:436.5Ref: TM-T17033
1mg69,00€5mg156,00€10mg225,00€25mg375,00€50mg533,00€100mg723,00€200mg938,00€1mL*10mM (DMSO)170,00€Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Fórmula:C15H21ClN6Pureza:98.60% - 98.92%Forma y color:SolidPeso molecular:320.82Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Fórmula:C13H12N2OPureza:98.29% - 99.92%Forma y color:Off-White SolidPeso molecular:212.258-Hydroxy-DPAT hydrobromide
CAS:8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Fórmula:C16H26BrNOPureza:98.90% - 99.09%Forma y color:SolidPeso molecular:328.29Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Forma y color:SolidPeso molecular:395.43CP94253 hydrochloride
CAS:CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Fórmula:C15H20ClN3OPureza:99.39%Forma y color:SolidPeso molecular:293.79Ref: TM-T22689
5mg70,00€10mg96,00€25mg216,00€50mg354,00€100mg567,00€200mg787,00€1mL*10mM (DMSO)70,00€Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Fórmula:C18H19ClN4Pureza:99.91% - 99.93%Forma y color:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecular:326.82Ref: TM-T0455
1g449,00€10mg35,00€25mg52,00€50mg70,00€100mg96,00€200mg170,00€500mg303,00€1mL*10mM (DMSO)47,00€L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Fórmula:C20H21N5O3SPureza:98.36%Forma y color:White SolidPeso molecular:411.48Naftopidil dihydrochloride
CAS:Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Fórmula:C24H28N2O3·2HClPureza:99.76%Forma y color:White SolidPeso molecular:465.41Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Fórmula:C8H11N5Pureza:99.54%Forma y color:SolidPeso molecular:177.21LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Fórmula:C27H23ClF4N4O3Pureza:98%Forma y color:SolidPeso molecular:562.94Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Fórmula:C25H27N3O2S·xHClPureza:99.05%Forma y color:SolidPeso molecular:433.6Ref: TM-T8690
1mg131,00€5mg286,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€500mg2.688,00€1mL*10mM (DMSO)338,00€S 16924
CAS:S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Fórmula:C22H24FNO4Pureza:98.23% - 99.45%Forma y color:SolidPeso molecular:385.43Methamnetamine hydrochloride
CAS:Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.Fórmula:C14H18ClNForma y color:SolidPeso molecular:235.75Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Fórmula:C19H24N2OPureza:98%Forma y color:SolidPeso molecular:296.41Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Fórmula:C14H15F3N6OPureza:97.63%Forma y color:SolidPeso molecular:340.3SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Fórmula:C32H33ClN4O3Pureza:97.82% - 98.09%Forma y color:SolidPeso molecular:557.085-HT2A receptor agonist-3
CAS:5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Fórmula:C21H26BrNO3Pureza:98%Forma y color:SolidPeso molecular:420.34
