Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Donitriptan hydrochloride
CAS:Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectivelyFórmula:C23H26ClN5O2Pureza:99.8% - 99.8%Forma y color:SolidPeso molecular:439.94Ref: TM-T21666
2mg40,00€5mg49,00€10mg64,00€25mg135,00€50mg240,00€100mg339,00€200mg439,00€500mgA consultarSumatriptan succinate
CAS:Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Fórmula:C18H27N3O6SPureza:97.53% - 99.51%Forma y color:White PowderPeso molecular:413.49Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Fórmula:C20H20ClNO4Pureza:99.79%Forma y color:SolidPeso molecular:373.8rac Desmethyl Citalopram Hydrochloride
CAS:rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.Fórmula:C19H20ClFN2OPureza:96.14%Forma y color:SolidPeso molecular:346.83Tegaserod
CAS:Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Fórmula:C16H23N5OPureza:99.89%Forma y color:SolidPeso molecular:301.39Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.5%Forma y color:SolidPeso molecular:492.68PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Pureza:98%Forma y color:Odour SolidAlprenolol
CAS:Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1AFórmula:C15H23NO2Pureza:99.73% - 99.78%Forma y color:SolidPeso molecular:249.35Mebhydrolin napadisylate
CAS:Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.77%Forma y color:White Or Almost White CrystallinePeso molecular:420.52Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Fórmula:C15H20ClN3O2·HClPureza:98.32%Forma y color:SolidPeso molecular:346.26Ref: TM-T5336
1mg46,00€5mg87,00€10mg144,00€25mg283,00€50mg454,00€100mg655,00€200mg930,00€1mL*10mM (DMSO)97,00€Protriptyline hydrochloride
CAS:Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.Fórmula:C19H21N·HClPureza:98.54% - 99.98%Forma y color:SolidPeso molecular:299.84Sulamserod
CAS:Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular relatedFórmula:C19H28ClN3O5SPureza:98.76%Forma y color:SolidPeso molecular:445.965-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Fórmula:C22H29FN4O2Pureza:99.25%Forma y color:SolidPeso molecular:400.49Ref: TM-T12597
1mg678,00€5mg1.359,00€10mg1.833,00€25mg2.727,00€50mg3.676,00€100mg4.969,00€1mL*10mM (DMSO)1.605,00€Lumateperone
CAS:Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Fórmula:C24H28FN3OPureza:99.77%Forma y color:SolidPeso molecular:393.5Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Fórmula:C22H20ClN3Pureza:99% - 99.66%Forma y color:SolidPeso molecular:361.87Masupirdine mesylate
CAS:Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's diseaseFórmula:C23H32BrN3O9S3Pureza:99.48%Forma y color:SolidPeso molecular:670.61Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Fórmula:C18H20N4Pureza:99.15%Forma y color:SolidPeso molecular:292.38SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFórmula:C15H14N4OPureza:99.61%Forma y color:SolidPeso molecular:266.3Ref: TM-T8357
1mg97,00€2mg150,00€5mg207,00€10mg311,00€25mg525,00€50mg757,00€100mg1.035,00€1mL*10mM (DMSO)216,00€AVN 322 free base
CAS:AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.Fórmula:C17H19N5O2SPureza:99.13%Forma y color:SolidPeso molecular:357.435-HT2A&5-HT2C agonist-1
CAS:5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.Fórmula:C14H20N2OPureza:98%Forma y color:SolidPeso molecular:232.32
