Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Dapoxetine
CAS:Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Fórmula:C21H23NOPureza:99.73%Forma y color:White To Off-White Crystalline PowderPeso molecular:305.42Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Fórmula:C23H24FN3O2SPureza:99.78%Forma y color:SolidPeso molecular:425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Fórmula:C50H68F2N6O4·C4H6O6Pureza:100% - 99.98%Forma y color:SolidPeso molecular:1005.2Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Fórmula:C21H21ClN4OSPureza:100% - 99.53%Forma y color:Tan SolidPeso molecular:412.94GM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Fórmula:C30H33FN2O4Forma y color:SolidPeso molecular:504.59Anpirtoline hydrochloride
CAS:Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Fórmula:C10H14Cl2N2SPureza:100% - 100%Forma y color:SolidPeso molecular:265.20Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:100% - 99.59%Forma y color:White Crystalline SolidPeso molecular:883.09Agomelatine
CAS:Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Fórmula:C15H17NO2Pureza:99.92%Forma y color:White SolidPeso molecular:243.3Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFórmula:C22H25N5O2Pureza:99% - 99.72%Forma y color:White To Off-White Crystalline PowderPeso molecular:391.47Ref: TM-T1512
10mg47,00€25mg79,00€50mg126,00€100mg183,00€200mg273,00€500mg462,00€1mL*10mM (DMSO)50,00€Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Forma y color:SolidPeso molecular:417.97RS-127445 hydrochloride
CAS:RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Fórmula:C17H17ClFN3Pureza:99.48%Forma y color:SolidPeso molecular:317.795-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFórmula:C17H22Cl2N6SPureza:98%Forma y color:SolidPeso molecular:413.37Paliperidone
CAS:Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Fórmula:C23H27FN4O3Pureza:95% - 99.08%Forma y color:Off White To Light Orange Coloured SolidPeso molecular:426.48Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Fórmula:C14H19ClN4O2Pureza:98%Forma y color:SolidPeso molecular:310.78(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Fórmula:C17H19N3Pureza:99.75%Forma y color:SolidPeso molecular:265.35Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Fórmula:C25H29N3O2Pureza:99.7% - 99.83%Forma y color:SolidPeso molecular:403.52F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Fórmula:C19H21ClF2N4OPureza:98.72%Forma y color:SolidPeso molecular:394.85Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFórmula:C28H33ClN2·2HClPureza:98.05%Forma y color:Off-White PowderPeso molecular:505.95idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Fórmula:C20H19F5N2OPureza:99.73%Forma y color:SolidPeso molecular:398.37Ref: TM-T7103
1mg88,00€2mg118,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€1mL*10mM (DMSO)187,00€Org 13011
CAS:Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Fórmula:C18H25F3N4OPureza:98.98%Forma y color:SoildPeso molecular:370.41Ref: TM-T28258L
1mg185,00€5mg459,00€10mg657,00€25mg1.026,00€50mg1.415,00€100mg1.872,00€1mL*10mM (DMSO)469,00€
