Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Fórmula:C19H27N3OPureza:99.52%Forma y color:SolidPeso molecular:313.44(±)-Fabesetron hydrochloride
CAS:FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.Fórmula:C18H20ClN3OPureza:98%Forma y color:SolidPeso molecular:329.82PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.Fórmula:C14H17ClN2OPureza:99.64%Forma y color:SolidPeso molecular:264.75SB-616234-A
CAS:SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.Fórmula:C32H36ClN5O3Pureza:99.68%Forma y color:SolidPeso molecular:574.11Ref: TM-T12847
1mg105,00€5mg255,00€10mg368,00€25mg557,00€50mg752,00€100mg1.035,00€200mg1.396,00€1mL*10mM (DMSO)321,00€5-HT2A/5-HT2C inverse agonist 1
CAS:5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A and 5-HT2C receptors, with hERG inhibition properties that mitigate cardiovascular risks. Demonstrating significant antipsychotic efficacy in the MK-801-induced mouse model, this compound holds potential for psychosis research.Fórmula:C24H35N5O2Forma y color:SolidPeso molecular:425.57Lofepramine
CAS:Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.Fórmula:C26H27ClN2OPureza:98.38%Forma y color:Crystals From Methanol Or Acetone SolidPeso molecular:418.96Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Forma y color:White SolidPeso molecular:414.43Ref: TM-T6493
1g283,00€10mg39,00€25mg55,00€50mg66,00€100mg90,00€200mg125,00€500mg197,00€1mL*10mM (DMSO)44,00€SB-399885 hydrochloride
CAS:SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.Fórmula:C18H22Cl3N3O4SPureza:98%Forma y color:SolidPeso molecular:482.81CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Fórmula:C15H18Cl2N4OPureza:99.50%Forma y color:SolidPeso molecular:341.24Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Fórmula:C20H26ClNO2Pureza:99.48%Forma y color:SolidPeso molecular:347.88Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Fórmula:C17H25N3O2SPureza:99.85%Forma y color:Light Yellow Or White PowerPeso molecular:335.462-Methyl-5-HT hydrochloride
CAS:2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Fórmula:C11H15ClN2OPureza:98%Forma y color:SolidPeso molecular:226.7(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Fórmula:C17H19N3Pureza:99.37%Forma y color:SolidPeso molecular:265.35AS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Fórmula:C18H25N3Pureza:98%Forma y color:SolidPeso molecular:283.41CP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."Fórmula:C29H21FN4OSPureza:97.81% - 99.11%Forma y color:SoildPeso molecular:492.57Nelotanserin
CAS:Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Fórmula:C18H15BrF2N4O2Pureza:98.01% - 98.42%Forma y color:SolidPeso molecular:437.24Ref: TM-T7350
1mg40,00€2mg52,00€5mg88,00€10mg119,00€25mg188,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)85,00€Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Forma y color:SolidPeso molecular:369.5Ref: TM-T2278
1mg40,00€2mg52,00€5mg88,00€10mg125,00€25mg233,00€50mg424,00€100mg613,00€500mg1.264,00€1mL*10mM (DMSO)127,00€2,6-DMA hydrochloride
CAS:2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Fórmula:C11H18ClNO2Forma y color:SolidPeso molecular:231.72Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Fórmula:C26H28FN3O9Pureza:99.68%Forma y color:SolidPeso molecular:545.51Paynantheine
CAS:Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Fórmula:C23H28N2O4Forma y color:SolidPeso molecular:396.48
