Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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ECPLA
CAS:ECPLA is an LSD analog and a potent 5-HT2A agonist (EC50 of 14.6 nM), capable of stimulating Gq-mediated calcium flux. It exhibits high affinity for most serotonin receptors, α2-adrenergic receptors, and D2-like dopamine receptors.Fórmula:C21H25N3OForma y color:SolidPeso molecular:335.44AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Fórmula:C23H31ClN2O2Pureza:99.14%Forma y color:SolidPeso molecular:402.96Ref: TM-T26543
1mg52,00€2mg74,00€5mg96,00€10mg137,00€25mg215,00€50mg391,00€100mg582,00€1mL*10mM (DMSO)127,00€Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.Fórmula:C16H20ClNOPureza:98.98% - 99.19%Forma y color:SoildPeso molecular:277.79Ref: TM-T67956L
1mg97,00€5mg217,00€10mg325,00€25mg557,00€50mg797,00€100mg1.103,00€1mL*10mM (DMSO)208,00€Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Fórmula:C21H20ClNO5Pureza:99.28%Forma y color:SolidPeso molecular:401.84Ref: TM-T1951
5mg35,00€10mg51,00€25mg80,00€50mg96,00€100mg135,00€200mg225,00€500mg373,00€1mL*10mM (DMSO)55,00€RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.Fórmula:C17H16FN3Pureza:99.32%Forma y color:SolidPeso molecular:281.33AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Fórmula:C17H21N5O2SPureza:99.81%Forma y color:SolidPeso molecular:359.45Ref: TM-T5179
1mg39,00€2mg49,00€5mg81,00€10mg120,00€25mg236,00€50mg354,00€100mg510,00€1mL*10mM (DMSO)89,00€Befiradol hydrochloride
CAS:Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.Fórmula:C20H23Cl2F2N3OPureza:99.1%Forma y color:SolidPeso molecular:430.32Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:100% - 99.93%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Fórmula:C27H26FN3OSPureza:98.55%Forma y color:SolidPeso molecular:459.58AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Fórmula:C17H20ClN5O2SPureza:98.83%Forma y color:SolidPeso molecular:393.89BW 723C86
CAS:BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.Fórmula:C16H19ClN2OSPureza:99.35%Forma y color:SolidPeso molecular:322.85Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Fórmula:C12H15N3O2Pureza:98%Forma y color:SolidPeso molecular:233.27CI 169369
CAS:CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.Fórmula:C19H21ClN2SPureza:100%Forma y color:SoildPeso molecular:344.9Paroxetine hydrochloride
CAS:Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.Fórmula:C19H21ClFNO3Pureza:98% - 99.99%Forma y color:White Crystalline PowderPeso molecular:365.8265-HT2A receptor agonist-5
CAS:5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.Fórmula:C23H29N3OForma y color:SolidPeso molecular:363.5Cannabidiolic acid methyl ester
CAS:Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Fórmula:C23H32O4Forma y color:SolidPeso molecular:372.5Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Forma y color:White SolidPeso molecular:506.47Ref: TM-T3275
5mg47,00€10mg70,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€1mL*10mM (DMSO)77,00€LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFórmula:C21H22FN3OPureza:99.32%Forma y color:SolidPeso molecular:351.42CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Fórmula:C19H28ClN5OPureza:98.41%Forma y color:SolidPeso molecular:377.91Ref: TM-T22671
1mg48,00€5mg101,00€10mg170,00€25mg270,00€50mg386,00€100mg520,00€1mL*10mM (DMSO)158,00€4-fluoro MBZP
CAS:4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.Fórmula:C12H17FN2Forma y color:SolidPeso molecular:208.28
