AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Productos de "AChR"
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Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Fórmula:C21H21N3O2Pureza:99.9%Forma y color:SolidPeso molecular:347.41Ref: TM-T10961
1mg215,00€5mg426,00€10mg598,00€25mg889,00€50mg1.188,00€100mg1.605,00€1mL*10mM (DMSO)472,00€Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Fórmula:C24H26ClNO4Pureza:99.78%Forma y color:White SolidPeso molecular:427.92Rivastigmine tartrate
CAS:Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.Fórmula:C14H22N2O2·C4H6O6Pureza:98% - 99.66%Forma y color:White To Off-White PowderPeso molecular:400.43Methyllycaconitine citrate
CAS:Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.Fórmula:C43H58N2O17Pureza:98.03% - 98.91%Forma y color:SolidPeso molecular:874.92Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Fórmula:C21H28BrNO3Pureza:99.29%Forma y color:SolidPeso molecular:422.36Homatropine Methylbromide
CAS:Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.Fórmula:C17H24BrNO3Pureza:98.97%Forma y color:SolidPeso molecular:370.299-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Fórmula:C7H9N5Pureza:99.35% - 99.41%Forma y color:SolidPeso molecular:163.18Trihexyphenidyl hydrochloride
CAS:Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.Fórmula:C20H32ClNOPureza:99.65%Forma y color:SolidPeso molecular:337.927Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Fórmula:C11H16ClNOPureza:98.9%Forma y color:SolidPeso molecular:213.7Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Fórmula:C19H20ClFN2O2Pureza:98.88%Forma y color:SolidPeso molecular:362.83Ref: TM-T9771
1mg66,00€5mg145,00€10mg226,00€25mg408,00€50mg558,00€100mg787,00€200mg1.035,00€1mL*10mM (DMSO)160,00€Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Fórmula:C14H23N3OSPureza:99.61%Forma y color:SolidPeso molecular:281.42Ref: TM-T36640
2mg38,00€5mg55,00€10mg93,00€25mg165,00€50mg264,00€100mg420,00€200mg607,00€1mL*10mM (DMSO)60,00€Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Fórmula:C28H30N2O2Pureza:99.78%Forma y color:SolidPeso molecular:426.55BQCA
CAS:BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.Fórmula:C18H15NO4Pureza:97.22%Forma y color:SolidPeso molecular:309.32Tematropium
CAS:Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.Fórmula:C21H31NO8SPureza:98.87%Forma y color:SolidPeso molecular:457.54Ref: TM-T10732
1mg212,00€2mg284,00€5mg449,00€10mg615,00€25mg929,00€50mg1.244,00€100mg1.691,00€1mL*10mM (DMSO)507,00€Tiotropium bromide
CAS:Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).Fórmula:C19H22BrNO4S2Pureza:96.82% - 99.63%Forma y color:White SolidPeso molecular:472.42Propoxur
CAS:Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.Fórmula:C11H15NO3Pureza:98.15% - 99.87%Forma y color:Minute Crystals (Niosh 2016)Peso molecular:209.24Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Fórmula:C22H32BrNO5Pureza:98.85%Forma y color:SolidPeso molecular:470.4Ref: TM-T28827
1mg74,00€5mg160,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€1mL*10mM (DMSO)170,00€Tribendimidine
CAS:Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.Fórmula:C28H32N6Pureza:≥98%Forma y color:SolidPeso molecular:452.59Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Fórmula:C29H34BrNO2Pureza:98.40% - 99.09%Forma y color:SolidPeso molecular:508.49Ref: TM-T4997
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg212,00€50mg350,00€100mg525,00€1mL*10mM (DMSO)87,00€VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Fórmula:C17H12F3NO4Pureza:100%Forma y color:SolidPeso molecular:351.28Ref: TM-T8007
2mg35,00€5mg52,00€10mg86,00€25mg144,00€50mg227,00€100mg359,00€500mg838,00€1mL*10mM (DMSO)58,00€
