AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Productos de "AChR"
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Emraclidine
CAS:Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.Fórmula:C20H21F3N4OPureza:99.84%Forma y color:SolidPeso molecular:390.4Ref: TM-T9694
1mg127,00€5mg305,00€10mg550,00€25mg882,00€50mg1.206,00€100mg1.605,00€1mL*10mM (DMSO)338,00€Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Fórmula:C19H23N3O3Pureza:99.96%Forma y color:SolidPeso molecular:341.4A 582941 HCl (848591-90-2(free base))
A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing propertiesFórmula:C17H21ClN4Pureza:99.83%Forma y color:SolidPeso molecular:316.83Ref: TM-T8725
1mg88,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)170,00€Orphenadrine Citrate
CAS:Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.Fórmula:C18H23NO·C6H8O7Pureza:98% - 99.51%Forma y color:White SolidPeso molecular:461.54BP-TQS
CAS:4BP-TQS is an allosteric agonist of α7 nAChRs.Fórmula:C18H17BrN2O2SPureza:99.96%Forma y color:SolidPeso molecular:405.31α-Muricholic acid
CAS:α-Muricholic acid is the most abundant primary bile acid in rodents.Fórmula:C24H40O5Pureza:98%Forma y color:SolidPeso molecular:408.57Succinylcholine Chloride Dihydrate
CAS:Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Forma y color:White SolidPeso molecular:397.34Propantheline bromide
CAS:Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscleFórmula:C23H30BrNO3Pureza:95% - ≥98%Peso molecular:448.4ML380
CAS:ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).Fórmula:C23H25F3N4O3SPureza:99.69%Forma y color:SolidPeso molecular:494.53Ref: TM-T28069
2mg49,00€5mg74,00€10mg119,00€25mg188,00€50mg354,00€100mg528,00€500mg1.159,00€1mL*10mM (DMSO)82,00€(-)-(S)-B-973B
CAS:(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.Fórmula:C24H26F2N6OPureza:99.52%Forma y color:SolidPeso molecular:452.5GP531
CAS:GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.Fórmula:C16H21N5O4Forma y color:SolidPeso molecular:347.37Cevimeline hydrochloride hemihydrate
CAS:Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.Fórmula:C20H38Cl2N2O3S2Pureza:98%Forma y color:SolidPeso molecular:489.55Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Fórmula:C12H17ClN2OPureza:99.23%Forma y color:SolidPeso molecular:240.729Ref: TM-T12201
5mg48,00€10mg71,00€25mg108,00€50mg160,00€100mg226,00€200mg331,00€1mL*10mM (DMSO)50,00€VU 0365114
CAS:VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).Fórmula:C22H14F3NO3Pureza:97.29%Forma y color:SolidPeso molecular:397.35Ref: TM-T13325
2mg38,00€5mg58,00€10mg82,00€25mg137,00€50mg224,00€100mg335,00€200mg469,00€1mL*10mM (DMSO)65,00€Tazomeline
CAS:Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.Fórmula:C14H23N3S2Pureza:100%Forma y color:SolidPeso molecular:297.48Oxyphencyclimine Hydrochloride
CAS:Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Fórmula:C20H29ClN2O3Pureza:99.55%Forma y color:SolidPeso molecular:380.91SIB 1553A
CAS:SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.Fórmula:C13H19NOSPureza:99.64%Forma y color:SoildPeso molecular:237.36Ref: TM-T16881L
1mg185,00€5mg459,00€10mg657,00€25mg1.026,00€50mg1.415,00€100mg1.872,00€1mL*10mM (DMSO)47,00€Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Fórmula:C20H24N·CH3O4SPureza:98% - 99.27%Forma y color:SolidPeso molecular:389.51Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Fórmula:C10H17IN2O2Pureza:98.93%Forma y color:SolidPeso molecular:324.16Ref: TM-T25538
1mg50,00€5mg107,00€10mg187,00€25mg411,00€50mg613,00€100mg873,00€500mg1.768,00€1mL*10mM (DMSO)117,00€Soclenicant
CAS:Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availabilityFórmula:C24H26N4O3Pureza:99.57%Forma y color:SoildPeso molecular:418.49Ref: TM-T203814
1mg201,00€5mg497,00€10mg701,00€25mg1.094,00€50mg1.508,00€100mg1.931,00€200mg2.637,00€
