AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Productos de "AChR"
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Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Fórmula:C23H26N2O2Pureza:99.87%Forma y color:SolidPeso molecular:362.46Vecuronium bromide
CAS:Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscleFórmula:C34H57BrN2O4Pureza:99.63% - 99.92%Forma y color:White PowderPeso molecular:637.73VU0453595
CAS:VU0453595 is a M1 positive allosteric modulator (PAM).Fórmula:C18H15FN4OPureza:99.48%Forma y color:SolidPeso molecular:322.34Lupinine
CAS:Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.Fórmula:C10H19NOPureza:99.95%Forma y color:SolidPeso molecular:169.26Ref: TM-FR16605
1mg95,00€5mg180,00€10mg271,00€25mg462,00€50mg672,00€100mg918,00€500mg1.840,00€1ml*10 (DMSO)151,00€Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.92%Forma y color:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Atropine methyl bromide
CAS:Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.Fórmula:C18H26BrNO3Pureza:99.70%Forma y color:SolidPeso molecular:384.308Ref: TM-T14345
1mg35,00€5mg70,00€10mg105,00€25mg187,00€50mg274,00€100mg404,00€200mg587,00€1mL*10mM (DMSO)77,00€Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Fórmula:C16H20N2O2Pureza:98.63%Forma y color:SolidPeso molecular:272.34Ref: TM-T22380
1mg93,00€2mg126,00€5mg187,00€10mg283,00€25mg462,00€50mg645,00€100mg867,00€200mg1.159,00€1mL*10mM (DMSO)187,00€Zamifenacin fumarate
CAS:Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.Fórmula:C31H33NO7Pureza:99.78%Forma y color:SolidPeso molecular:531.6Ref: TM-T13385
1mg40,00€5mg88,00€10mg119,00€25mg216,00€50mg354,00€100mg533,00€200mg743,00€1mL*10mM (DMSO)93,00€RPR121056
CAS:RPR121056 is a Irinotecan metabolite, which is generated by CYP3A4. Irinotecan is an antineoplastic agent that inhibits topoisomerase type I.Fórmula:C33H38N4O8Pureza:98%Forma y color:SolidPeso molecular:618.68GSK-1034702
CAS:GSK-1034702 is an M1 mAChR agonist that improves cognitive deficits and may be useful in the study of neurologic disorders.Fórmula:C18H24FN3O2Pureza:99.69%Forma y color:SolidPeso molecular:333.4Sch412348
CAS:Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.Fórmula:C22H21F2N9OPureza:98%Forma y color:SolidPeso molecular:465.46Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Fórmula:C9H12Cl2N2OPureza:95% - 98.71%Forma y color:SolidPeso molecular:235.11(Rac)-Sabcomeline
CAS:(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.Fórmula:C10H15N3OPureza:99.14%Forma y color:SolidPeso molecular:193.25Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Fórmula:C18H17N3O3SPureza:98.46%Forma y color:SolidPeso molecular:355.41GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Fórmula:C19H20N2O2Pureza:98%Forma y color:SolidPeso molecular:308.37TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.Fórmula:C25H32N4OPureza:97.87% - 99.9%Forma y color:SolidPeso molecular:404.55NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Fórmula:C27H44ClNO8Pureza:98% - 98%Forma y color:SolidPeso molecular:546.09TZ3O
CAS:TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type model in rats.Fórmula:C18H13NO4SPureza:99.84%Forma y color:SolidPeso molecular:339.37Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.50%Forma y color:SolidPeso molecular:359.89
