AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Productos de "AChR"
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bPiDDB
CAS:bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.Fórmula:C24H38Br2N2Pureza:98.72%Forma y color:SolidPeso molecular:514.38Ref: TM-T37818
2mg43,00€5mg60,00€10mg96,00€25mg188,00€50mg278,00€100mg411,00€200mg607,00€1mL*10mM (DMSO)73,00€Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Forma y color:SolidPeso molecular:552.7Loxeen
CAS:Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.Fórmula:C20H25NO·CH4O3SPureza:99.46%Forma y color:White To Off-White Crystalline PowderPeso molecular:391.52Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Fórmula:C24H31N5O2Pureza:99.81%Forma y color:SolidPeso molecular:421.54Cimetropium Bromide
CAS:Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.Fórmula:C21H28BrNO4Forma y color:SolidPeso molecular:438.36Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Fórmula:C17H17N5O6SPureza:98.83% - 99.69%Forma y color:Off-White SolidPeso molecular:419.414-DAMP
CAS:4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.Fórmula:C21H26INO2Pureza:98%Forma y color:SolidPeso molecular:451.34Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Fórmula:C20H21N3OPureza:99.17%Forma y color:SolidPeso molecular:319.4Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Fórmula:C22H31NOPureza:99.71%Forma y color:White Like Or Light Brown Crystalline PowderPeso molecular:325.49Mepenzolate Bromide
CAS:Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.Fórmula:C21H26BrNO3Pureza:95.73% - 99.21%Forma y color:SolidPeso molecular:420.34Aclidinium bromide
CAS:Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.Fórmula:C26H30NO4S2·BrPureza:98.93% - 99.69%Forma y color:SolidPeso molecular:564.55Ref: TM-T2555
2mg39,00€5mg57,00€10mg88,00€25mg145,00€50mg234,00€100mg350,00€500mg825,00€1mL*10mM (DMSO)72,00€Clidinium bromide
CAS:Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.Fórmula:C22H26BrNO3Pureza:98.89% - 99.86%Forma y color:White Crystalline SolidPeso molecular:432.35SQ22536
CAS:SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.Fórmula:C9H11N5OPureza:99.18%Forma y color:Off-White SolidPeso molecular:205.22SCH-900271
CAS:SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.Fórmula:C14H16N2O4Pureza:98.25% - 99%Forma y color:SolidPeso molecular:276.29Ref: TM-T34573
1mg118,00€5mg275,00€10mg419,00€25mg692,00€50mg938,00€100mg1.320,00€500mg2.632,00€1mL*10mM (DMSO)263,00€Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Fórmula:C23H27ClN2O2Pureza:99.32%Forma y color:Off-White PowderPeso molecular:398.93Oxitropium Bromide
CAS:Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.Fórmula:C19H26BrNO4Pureza:98%Forma y color:SolidPeso molecular:412.32Nanofin
CAS:Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.Fórmula:C7H15NPureza:99.818%Forma y color:Clear Colorless To Slightly Yellow LiquidPeso molecular:113.2AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Fórmula:C27H38N6O2Pureza:98%Forma y color:SolidPeso molecular:478.63TAK-071
CAS:TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).Fórmula:C24H24FN3O3Pureza:98.02%Forma y color:SolidPeso molecular:421.46Carbachol
CAS:Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.Fórmula:C6H15ClN2O2Pureza:100% - 90%Forma y color:SolidPeso molecular:182.65
