NMDAR
Los inhibidores del receptor de N-Metil-D-Aspartato (NMDAR) son compuestos que bloquean la actividad de los NMDARs, un subtipo de receptores de glutamato que desempeñan un papel crítico en la plasticidad sináptica, el aprendizaje y la memoria. La sobreactivación de los NMDARs está implicada en la excitotoxicidad, que puede llevar a daño neuronal y está asociada con condiciones como el accidente cerebrovascular, el trauma craneoencefálico y enfermedades neurodegenerativas. Los inhibidores de NMDAR son herramientas esenciales para estudiar la excitotoxicidad y para desarrollar terapias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de NMDAR para apoyar su investigación en función sináptica, neuroprotección y trastornos cognitivos.
Productos de "NMDAR"
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AV-101
CAS:AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.Fórmula:C10H11ClN2O3Pureza:97.84% - 98.27%Forma y color:SolidPeso molecular:242.66BZAD01
CAS:BZAD01 is a selective NMDA NR1A/2B receptor antagonist.Fórmula:C16H12F6N2OPureza:99.51% - 99.78%Forma y color:SolidPeso molecular:362.27Ref: TM-T25196
5mg50,00€10mg84,00€25mg150,00€50mg226,00€100mg375,00€200mg523,00€1mL*10mM (DMSO)71,00€Aptiganel
CAS:Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.Fórmula:C20H21N3Pureza:98.19% - 98.90%Forma y color:SolidPeso molecular:303.4Delucemine Hydrochloride
CAS:Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.Fórmula:C16H18ClF2NPureza:98.14% - 99.53%Forma y color:SolidPeso molecular:297.77Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Fórmula:C10H14O3Pureza:99.49%Forma y color:SolidPeso molecular:182.22ZL006
CAS:ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Fórmula:C14H11Cl2NO4Pureza:98.29%Forma y color:SolidPeso molecular:328.15Ref: TM-T17293
5mg50,00€10mg66,00€25mg117,00€50mg180,00€100mg306,00€200mg444,00€1mL*10mM (DMSO)52,00€(-)-Dizocilpine maleate
CAS:(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.Fórmula:C20H19NO4Pureza:99.89%Forma y color:White SolidPeso molecular:337.37RPR104632
CAS:RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective activity.Fórmula:C15H11BrCl2N2O4SPureza:99.06%Forma y color:SolidPeso molecular:466.13Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Fórmula:C13H18ClNO2Pureza:98.51% - 98.64%Forma y color:SolidPeso molecular:255.74Dizocilpine
CAS:MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.Fórmula:C16H15NPureza:99.75% - 99.97%Forma y color:SolidPeso molecular:221.3MDL-29951
CAS:MDL-29951 is a novel glycine antagonist of NMDA receptor activation.Fórmula:C12H9Cl2NO4Pureza:99.07% - 99.49%Forma y color:SolidPeso molecular:302.11Ref: TM-T1897
1mg50,00€5mg104,00€10mg180,00€25mg325,00€50mg469,00€100mg645,00€200mg868,00€1mL*10mM (DMSO)108,00€Gacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Fórmula:C16H25NSPureza:100% - 99%Forma y color:SolidPeso molecular:263.44BDBM50597431
CAS:BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's disease and Parkinson's syndrome.Fórmula:C27H43F3O2Pureza:98.64% - 99.28%Forma y color:SoildPeso molecular:456.62ALDH3A1-IN-1
CAS:ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with IC50 of 1.61 μM, outperforms DEAB in prostate cancer cells.Fórmula:C13H18N2O3Pureza:99.86%Forma y color:SolidPeso molecular:250.29Ro 25-6981
CAS:Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.Fórmula:C22H29NO2Pureza:99.44%Forma y color:SolidPeso molecular:339.47L-Cysteine S-sulfate
CAS:L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.Fórmula:C3H7NO5S2Pureza:98.92% - 99.92%Forma y color:SolidPeso molecular:201.22PEAQX
CAS:PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).Fórmula:C17H17BrN3O5PPureza:100% - ≥98%Forma y color:SolidPeso molecular:454.21Ref: TM-T4171
1mg34,00€2mg46,00€5mg74,00€10mg125,00€25mg216,00€50mg338,00€100mg470,00€200mg680,00€1mL*10mM (DMSO)97,00€Co 101244 hydrochloride
CAS:Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Fórmula:C21H28ClNO3Pureza:98.44%Forma y color:SolidPeso molecular:377.9MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFórmula:C11H6BrN3O3Pureza:98.13%Forma y color:SolidPeso molecular:308.09Ref: TM-T12110
1mg96,00€5mg202,00€10mg329,00€25mg655,00€50mg1.103,00€100mg1.483,00€1mL*10mM (DMSO)224,00€Rapastinel
CAS:Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.Fórmula:C18H31N5O6Pureza:97.18%Forma y color:SolidPeso molecular:413.47
