Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Fórmula:C17H21N5OPureza:100% - 99.67%Forma y color:SolidPeso molecular:311.38Dalcotidine
CAS:Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.Fórmula:C18H29N3O2Pureza:98.34%Forma y color:SolidPeso molecular:319.44Ref: TM-T31195
1mg94,00€5mg205,00€10mg303,00€25mg490,00€50mg710,00€100mg998,00€200mg1.349,00€1mL*10mM (DMSO)205,00€Acrivastine
CAS:Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Fórmula:C22H24N2O2Pureza:100% - 99.73%Forma y color:SolidPeso molecular:348.44Ref: TM-T4551
1g792,00€5mg37,00€10mg51,00€25mg99,00€50mg160,00€100mg221,00€500mg553,00€1mL*10mM (DMSO)40,00€Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Fórmula:C18H22ClNOPureza:99.44%Forma y color:SolidPeso molecular:303.83Fexofenadine hydrochloride
CAS:Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Fórmula:C32H39NO4·HClPureza:99.39% - ≥95%Forma y color:SolidPeso molecular:538.13Azelastine hydrochloride
CAS:Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.Fórmula:C22H24ClN3O·HClPureza:100% - 99.97%Forma y color:White Crystalline PowderPeso molecular:418.36Chloropyramine hydrochloride
CAS:Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.Fórmula:C16H20ClN3·HClPureza:99.45% - 99.8%Forma y color:SolidPeso molecular:326.26Dexchlorpheniramine Maleate
CAS:Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Fórmula:C20H23ClN2O4Pureza:99.58%Forma y color:White Or Almost White Crystalline PowderPeso molecular:390.86Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Fórmula:C17H19N3Pureza:99.98%Forma y color:SolidPeso molecular:265.35Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Fórmula:C16H21N3·HClPureza:100% - 99.54%Forma y color:White SolidPeso molecular:291.82KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Fórmula:C26H28N4O3Pureza:98.13%Forma y color:SoildPeso molecular:444.53H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Fórmula:C20H28F2N2OPureza:98%Forma y color:SolidPeso molecular:350.45PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Fórmula:C25H32F2N2O4SPureza:98%Forma y color:SolidPeso molecular:494.6Clobenpropit dihydrobromide
CAS:Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)Fórmula:C14H19Br2ClN4SPureza:99.86%Forma y color:SolidPeso molecular:470.7Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Fórmula:C9H16N4S2Pureza:97.41%Forma y color:SolidPeso molecular:244.38Bromodiphenhydramine hydrochloride
CAS:Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.Fórmula:C17H21BrClNOPureza:97.31%Forma y color:SolidPeso molecular:370.71UR-AK49
CAS:UR-AK49 (compound 11) is an agonist for the human histamine H1 and H2 receptors. It exhibits an EC50 of 23 nM in the GTPase assay involving hH2R-Gsalpha fusion protein expressed in Sf9 insect cells. UR-AK49 is applicable in neurologically related research.Fórmula:C16H27N5OForma y color:SolidPeso molecular:305.42Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Fórmula:C21H28N2O5Pureza:99.61%Forma y color:5 1 (Ntp 1992)Peso molecular:388.46MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).Fórmula:C23H24F3N3O2Pureza:99.79%Forma y color:SolidPeso molecular:431.45Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Fórmula:C18H20N2Pureza:99.39%Forma y color:SolidPeso molecular:264.36
