
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Forma y color:SolidPeso molecular:458.42Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Fórmula:C15H20Cl2N2O3Pureza:99.17%Forma y color:SolidPeso molecular:347.24MPTP hydrochloride
CAS:MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.Fórmula:C12H16ClNPureza:100% - 99.73%Forma y color:SolidPeso molecular:209.72Ref: TM-T4081
1g758,00€5mg35,00€10mg52,00€25mg87,00€50mg145,00€100mg197,00€200mg313,00€500mg527,00€1mL*10mM (DMSO)55,00€MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Fórmula:C24H23N3O2Pureza:99.85%Forma y color:SolidPeso molecular:385.46L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Fórmula:C18H22Cl4N4Pureza:97.52%Forma y color:SolidPeso molecular:436.21Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Fórmula:C21H33Cl3N4OPureza:100% - 98.52%Forma y color:SolidPeso molecular:463.87Desipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Fórmula:C18H23ClN2Pureza:99.58% - 99.94%Forma y color:White To Off-White PowderPeso molecular:302.842BisfluoroModafinil
CAS:CRL-40940 is a selective dopaminergic reuptake inhibitorFórmula:C15H13F2NO2SPureza:99.19%Forma y color:SolidPeso molecular:309.33Ref: TM-T4262
1mg48,00€2mg64,00€5mg94,00€10mg139,00€25mg236,00€50mg359,00€100mg540,00€500mg1.130,00€1mL*10mM (DMSO)104,00€Zuclopenthixol
CAS:Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.Fórmula:C22H25ClN2OSPureza:98.90% - 99.82%Forma y color:SolidPeso molecular:400.96Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Fórmula:C21H22ClFN4O2Pureza:96.29%Forma y color:SolidPeso molecular:416.88Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Fórmula:C10H17N3SPureza:99.78%Forma y color:SolidPeso molecular:211.33WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Fórmula:C25H34N4O2·C4H4O4Pureza:99.26% - 99.68%Forma y color:SolidPeso molecular:538.64Ref: TM-T2631
2mg46,00€5mg66,00€10mg95,00€25mg180,00€50mg334,00€100mg495,00€200mg717,00€500mg1.111,00€1mL*10mM (DMSO)79,00€Bromocriptine mesylate
CAS:Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Fórmula:C33H44BrN5O8SPureza:99.76% - 99.87%Forma y color:White SolidPeso molecular:750.7Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Fórmula:C23H30N4O2SPureza:99.23%Forma y color:White PowderPeso molecular:426.57Timiperone
CAS:Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it mitigates stereotyped behavior.Fórmula:C22H24FN3OSPureza:98%Forma y color:SolidPeso molecular:397.51Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Fórmula:C23H26N2OPureza:99.08% - 99.18%Forma y color:SolidPeso molecular:346.47Asenapine hydrochloride
CAS:Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Fórmula:C17H17Cl2NOForma y color:SolidPeso molecular:322.23SPD-473 citrate
CAS:SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Fórmula:C23H31Cl2NO8SPureza:99.37%Forma y color:SolidPeso molecular:552.475,7-Dimethoxyluteolin
CAS:5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator with an EC50 of 3.417 μM.Fórmula:C17H14O6Pureza:99.56% - 99.56%Forma y color:SolidPeso molecular:314.29WAY-100635
CAS:WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Fórmula:C25H34N4O2Forma y color:SolidPeso molecular:422.56