Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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Didesmethyl cariprazine
CAS:Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.Fórmula:C19H28Cl2N4OPureza:99.70%Forma y color:SolidPeso molecular:399.36L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Fórmula:C20H21ClN2OPureza:98.57%Forma y color:SolidPeso molecular:340.85Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Fórmula:C25H29N3O2Pureza:99.7% - 99.83%Forma y color:SolidPeso molecular:403.52Aripiprazole Lauroxil
CAS:Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Fórmula:C36H51Cl2N3O4Pureza:98.06%Forma y color:SolidPeso molecular:660.71Ref: TM-T14319
10mg48,00€25mg72,00€50mg96,00€100mg130,00€200mg188,00€500mg318,00€1mL*10mM (DMSO)49,00€Dihydrexidine
CAS:Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.Fórmula:C17H17NO2Pureza:98%Forma y color:SolidPeso molecular:267.32Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Fórmula:C15H17N5SPureza:98.93%Forma y color:SolidPeso molecular:299.39Ref: TM-T12405
1mg487,00€5mg753,00€10mg1.216,00€25mg1.691,00€50mg2.262,00€100mg3.068,00€1mL*10mM (DMSO)938,00€Domperidone
CAS:Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.Fórmula:C22H24ClN5O2Pureza:98% - 99.82%Forma y color:SolidPeso molecular:425.91DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Fórmula:C11H11Cl2NPureza:96.7%Forma y color:SolidPeso molecular:228.12Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Forma y color:SolidPeso molecular:643.71Eticlopride hydrochloride
CAS:Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Fórmula:C17H25ClN2O3·HClPureza:98%Forma y color:SolidPeso molecular:377.31Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Fórmula:C19H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:329.82Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Fórmula:C24H32N4O2SPureza:99.52%Forma y color:SolidPeso molecular:440.6Ref: TM-T24885
1mg130,00€5mg309,00€10mg567,00€25mg910,00€50mg1.225,00€100mg1.644,00€1mL*10mM (DMSO)374,00€Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Fórmula:C23H30FN3Pureza:99.85%Forma y color:SolidPeso molecular:367.5Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Fórmula:C14H22ClN3O2Pureza:99.75%Forma y color:SolidPeso molecular:299.8Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Fórmula:C8H12N2Pureza:98%Forma y color:LiquidPeso molecular:136.19Ref: TM-T9540
5mgA consultar10mgA consultar25mgA consultar50mgA consultar100mgA consultar200mgA consultar500mgA consultarBrilaroxazine
CAS:Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Fórmula:C22H25Cl2N3O3Pureza:98.00%Forma y color:SolidPeso molecular:450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Fórmula:C20H27F3N6OSPureza:98.62%Forma y color:SolidPeso molecular:456.53Ref: TM-T10213
1mg89,00€5mg198,00€10mg279,00€25mg434,00€50mg562,00€100mg780,00€200mg1.035,00€1mL*10mM (DMSO)227,00€Ecopipam
CAS:Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Fórmula:C19H20ClNOPureza:98.5%Forma y color:SolidPeso molecular:313.82Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Fórmula:C16H26N2O2Pureza:99.52%Forma y color:SolidPeso molecular:278.39LE 300
CAS:LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Fórmula:C20H22N2Pureza:98.08% - 98.35%Forma y color:SolidPeso molecular:290.4
