
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
Ordenar por
SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Fórmula:C21H22ClNO5Pureza:98%Forma y color:SolidPeso molecular:403.86Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Forma y color:White PowderPeso molecular:390.4Tetrahydropalmatine
CAS:Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epilepticFórmula:C21H25NO4Pureza:99.91% - 99.95%Forma y color:SolidPeso molecular:355.43FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].Fórmula:C33H36N4O2Pureza:98%Forma y color:SolidPeso molecular:520.66NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Fórmula:C28H29Cl2N3OPureza:98.79%Forma y color:SolidPeso molecular:494.46Ref: TM-T28167
2mg40,00€5mg58,00€10mg90,00€25mg163,00€50mg279,00€100mg394,00€500mgA consultar1mL*10mM (DMSO)75,00€PD 168568 dihydrochloride
CAS:PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Fórmula:C22H29Cl2N3OPureza:99.27%Forma y color:SolidPeso molecular:422.39Ref: TM-T12383
5mg48,00€10mg58,00€25mg117,00€50mg170,00€100mg248,00€200mg348,00€1mL*10mM (DMSO)60,00€Pimethixene maleate
CAS:Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Fórmula:C23H23NO4SPureza:100%Forma y color:SolidPeso molecular:409.5SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Fórmula:C17H19Cl2NOPureza:98% - 99.51%Forma y color:SolidPeso molecular:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€Ordopidine
CAS:Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.Fórmula:C14H20FNO2SPureza:99.52%Forma y color:SolidPeso molecular:285.38Spiroxatrine
CAS:Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Fórmula:C22H25N3O3Pureza:99.83%Forma y color:SolidPeso molecular:379.45D-tetrahydropalmatine
CAS:D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Fórmula:C21H25NO4Pureza:99.34%Forma y color:SolidPeso molecular:355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Fórmula:C17H27ClN2O4SPureza:≥95%Forma y color:White Or Yellowish PowderPeso molecular:390.93Droperidol
CAS:Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Fórmula:C22H22FN3O2Pureza:97.16% - 98%Forma y color:SolidPeso molecular:379.43Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Fórmula:C17H22Cl2N4Pureza:99.95%Forma y color:SolidPeso molecular:353.29Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Fórmula:C21H21ClN4OSPureza:100% - 99.53%Forma y color:Tan SolidPeso molecular:412.94Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:100% - 99.59%Forma y color:White Crystalline SolidPeso molecular:883.09Seridopidine
CAS:Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Fórmula:C14H20FNO2SPureza:99.11%Forma y color:SolidPeso molecular:285.38Bromopride
CAS:Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Fórmula:C14H22BrN3O2Pureza:99.95%Forma y color:SolidPeso molecular:344.25Ref: TM-T1175
2mg44,00€5mg65,00€10mg93,00€25mg178,00€50mg281,00€100mg454,00€200mg650,00€1mL*10mM (DMSO)71,00€CP-226269
CAS:CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.Fórmula:C18H19FN4Pureza:99.08%Forma y color:SolidPeso molecular:310.37Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Fórmula:C19H27NO3Pureza:98% - 99.91%Forma y color:White To Off-White White To Off-White SolidPeso molecular:317.42