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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Productos de "Receptor de dopamina"

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productos por página.Hay 309 productos en esta categoría.
  • L-745870 hydrochloride

    CAS:
    L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor
    Fórmula:C18H20Cl2N4
    Pureza:97.36%
    Forma y color:Solid
    Peso molecular:363.28

    Ref: TM-T11799

    5mg
    40,00€
    10mg
    65,00€
    25mg
    111,00€
    50mg
    178,00€
    100mg
    259,00€
    200mg
    374,00€
    1mL*10mM (DMSO)
    34,00€
  • Levosulpiride

    CAS:
    Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Forma y color:White Crystalline Powder
    Peso molecular:341.43

    Ref: TM-T1211

    100mg
    55,00€
    1mL*10mM (DMSO)
    55,00€
  • Diclofensine hydrochloride

    CAS:
    Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
    Fórmula:C17H18Cl3NO
    Pureza:98.86% - 99.93%
    Forma y color:Solid
    Peso molecular:358.69

    Ref: TM-T7745

    5mg
    51,00€
    10mg
    85,00€
    25mg
    153,00€
    50mg
    283,00€
    100mg
    406,00€
    200mg
    568,00€
  • FAUC 213

    CAS:
    FAUC 213 is a selective full antagonist of the dopamine D4 receptor.
    Fórmula:C18H19ClN4
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:326.82

    Ref: TM-T24055

    2mg
    39,00€
    5mg
    62,00€
    10mg
    87,00€
    25mg
    170,00€
    50mg
    A consultar
  • Nomifensine maleate

    CAS:
    Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
    Fórmula:C20H22N2O4
    Pureza:98.46%
    Forma y color:Solid
    Peso molecular:354.4

    Ref: TM-T7070

    10mg
    44,00€
    25mg
    65,00€
    50mg
    95,00€
    100mg
    155,00€
    1mL*10mM (DMSO)
    55,00€
  • Tolnapersine

    CAS:
    Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
    Fórmula:C21H26N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:322.44

    Ref: TM-T68023

    1mg
    126,00€
    5mg
    304,00€
    10mg
    447,00€
    25mg
    873,00€
    50mg
    1.188,00€
    100mg
    1.843,00€
  • Clozapine

    CAS:
    Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.
    Fórmula:C18H19ClN4
    Pureza:99.91% - 99.93%
    Forma y color:Yellow Crystals From Acetone-Petroleum Ether Solid
    Peso molecular:326.82

    Ref: TM-T0455

    1g
    449,00€
    10mg
    35,00€
    25mg
    52,00€
    50mg
    70,00€
    100mg
    96,00€
    200mg
    170,00€
    500mg
    303,00€
    1mL*10mM (DMSO)
    47,00€
  • Brexpiprazole HCl

    CAS:
    Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.
    Fórmula:C25H27N3O2S·xHCl
    Pureza:99.05%
    Forma y color:Solid
    Peso molecular:433.6

    Ref: TM-T8690

    1mg
    131,00€
    5mg
    286,00€
    10mg
    430,00€
    25mg
    710,00€
    50mg
    998,00€
    100mg
    1.349,00€
    500mg
    2.688,00€
    1mL*10mM (DMSO)
    338,00€
  • A-381393

    CAS:
    A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).
    Fórmula:C20H24N4
    Pureza:99.00%
    Forma y color:Solid
    Peso molecular:320.43

    Ref: TM-T5397

    1mg
    40,00€
    5mg
    80,00€
    10mg
    117,00€
    25mg
    210,00€
    50mg
    304,00€
    100mg
    437,00€
    200mg
    615,00€
    1mL*10mM (DMSO)
    88,00€
  • Hirsuteine

    CAS:
    Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.
    Fórmula:C22H26N2O3
    Pureza:99.36% - 99.63%
    Forma y color:Solid
    Peso molecular:366.45

    Ref: TM-TN1081

    1mg
    92,00€
    5mg
    187,00€
    10mg
    280,00€
    25mg
    472,00€
    50mg
    A consultar
    1mL*10mM (DMSO)
    200,00€
  • Pramipexole dihydrochloride

    CAS:
    Pramipexole dihydrochloride could be used to treat Parkinson disease.
    Fórmula:C10H18ClN3S
    Pureza:98%
    Forma y color:White Crystalline Powder
    Peso molecular:247.79

    Ref: TM-T1476L

    5mg
    35,00€
    10mg
    59,00€
  • D1R antagonist 1

    CAS:
    Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].
    Fórmula:C22H26BrNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:448.35

    Ref: TM-T78735

    1mg
    185,00€
    5mg
    459,00€
    10mg
    657,00€
    25mg
    1.026,00€
    50mg
    1.415,00€
    100mg
    1.872,00€
  • Tetrahydropalmatine hydrochloride

    CAS:
    Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.
    Fórmula:C21H26ClNO4
    Pureza:98% - 99.59%
    Forma y color:Solid
    Peso molecular:391.888

    Ref: TM-T2917

    25mg
    40,00€
    50mg
    51,00€
    100mg
    74,00€
    200mg
    97,00€
  • PF2562

    CAS:
    PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).
    Fórmula:C19H17N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:331.37

    Ref: TM-T16511

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • AHN 1-055 hydrochloride

    CAS:
    AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).
    Fórmula:C21H24ClF2NO
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:379.87

    Ref: TM-T39429

    2mg
    35,00€
    5mg
    52,00€
    10mg
    80,00€
    25mg
    137,00€
    50mg
    202,00€
    100mg
    311,00€
    200mg
    467,00€
    1mL*10mM (DMSO)
    52,00€
  • Talipexole dihydrochloride

    CAS:
    Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and
    Fórmula:C10H17Cl2N3S
    Pureza:98.64%
    Forma y color:Light Yellow Solid
    Peso molecular:282.23

    Ref: TM-T14490

    2mg
    38,00€
    5mg
    56,00€
    10mg
    89,00€
    25mg
    154,00€
    50mg
    264,00€
    100mg
    424,00€
    200mg
    613,00€
    500mg
    949,00€
    1mL*10mM (DMSO)
    63,00€
  • PNU-96391

    CAS:
    PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.
    Fórmula:C15H23NO2S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:281.41

    Ref: TM-T28435

    1mg
    115,00€
    5mg
    249,00€
    10mg
    369,00€
    25mg
    562,00€
    50mg
    787,00€
    100mg
    1.054,00€
    200mg
    1.406,00€
    1mL*10mM (DMSO)
    235,00€
  • Veralipride

    CAS:
    Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.
    Fórmula:C17H25N3O5S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:383.46

    Ref: TM-T7632

    1mg
    65,00€
    5mg
    139,00€
    10mg
    205,00€
    25mg
    378,00€
    50mg
    587,00€
    100mg
    882,00€
    1mL*10mM (DMSO)
    155,00€
  • N-0500 HCl

    CAS:
    N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
    Fórmula:C15H22ClNO2
    Pureza:98.3% - 98.42%
    Forma y color:Solid
    Peso molecular:283.79

    Ref: TM-T60107

    5mg
    35,00€
    10mg
    55,00€
  • SK609 HCl

    CAS:
    SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.
    Fórmula:C10H15Cl2N
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:220.14

    Ref: TM-T24797

    1mg
    88,00€
    5mg
    187,00€
    10mg
    274,00€
    25mg
    467,00€
    50mg
    652,00€
    100mg
    924,00€
    500mg
    1.833,00€