
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Fórmula:C20H29FN2O3Pureza:100% - 99.17%Forma y color:SolidPeso molecular:364.45Ref: TM-T70302
1mg359,00€5mg842,00€10mg1.035,00€25mg1.663,00€50mg2.072,00€100mg2.660,00€1mL*10mM (DMSO)677,00€Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Fórmula:C22H24ClN3O5Pureza:99.69%Forma y color:White To Of-White SolidPeso molecular:445.95-HT7R antagonist 3
CAS:Compound 6.4, also known as 5-HT7R antagonist 3, is a selective antagonist of the 5-HT7R with a Ki of 8 nM. It exhibits significantly less affinity towards D2R, 5-HT1AR, and 5-HT2AR with Ki values of 511 nM, 8930 nM, and 5786 nM, respectively. In mice, 5-HT7R antagonist 3 demonstrates anti-depressant and anti-anxiety activities.Fórmula:C30H33FN4O3Forma y color:SolidPeso molecular:516.61Pericyazine
CAS:Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.Fórmula:C21H23N3OSPureza:99.61%Forma y color:SolidPeso molecular:365.49Ref: TM-T16472
1mg46,00€2mg59,00€5mg93,00€10mg124,00€25mg235,00€50mg389,00€100mg567,00€500mg1.225,00€1mL*10mM (DMSO)77,00€Piribedil
CAS:Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.Fórmula:C16H18N4O2Pureza:99.79% - 99.91%Forma y color:SolidPeso molecular:298.34Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Fórmula:C23H24FN3O2SPureza:99.78%Forma y color:SolidPeso molecular:425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Fipexide
CAS:Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.Fórmula:C20H21ClN2O4Pureza:99.95%Forma y color:SolidPeso molecular:388.84Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.5%Forma y color:SolidPeso molecular:492.68(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Fórmula:C19H26ClNOSForma y color:SolidPeso molecular:351.93Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Fórmula:C24H36O2Forma y color:SolidPeso molecular:356.54Amantadine hydrochloride
CAS:Amantadine hydrochloride (CI-719) is an antiviral that is used in the prophylactic or symptomatic treatment of influenza A and Parkinson disease.Fórmula:C10H18ClNPureza:99.98%Forma y color:Solid CrystallinePeso molecular:187.71Sonepiprazole
CAS:Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine receptors, exhibiting dissociationFórmula:C21H27N3O3SPureza:99.31%Forma y color:SolidPeso molecular:401.52Ref: TM-T23380
2mg38,00€5mg58,00€10mg94,00€25mg180,00€50mg306,00€100mg442,00€200mg622,00€1mL*10mM (DMSO)71,00€UCM-1306
CAS:UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.Fórmula:C14H14FNO2SPureza:100%Forma y color:SoildPeso molecular:279.33Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Forma y color:SolidPeso molecular:417.97Paliperidone
CAS:Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Fórmula:C23H27FN4O3Pureza:95% - 99.08%Forma y color:Off White To Light Orange Coloured SolidPeso molecular:426.48Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Fórmula:C28H42F2N2O12S2Pureza:99.98%Forma y color:SolidPeso molecular:700.77Lumateperone
CAS:Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Fórmula:C24H28FN3OPureza:99.77%Forma y color:SolidPeso molecular:393.5Haloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Fórmula:C21H23ClFNO2Pureza:98.69% - 98.97%Forma y color:Crystals SolidPeso molecular:375.86Moperone
CAS:Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Fórmula:C22H26FNO2Forma y color:SolidPeso molecular:355.45PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Fórmula:C24H26N4O5Pureza:98.82%Forma y color:SolidPeso molecular:450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€