Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Forma y color:SolidPeso molecular:328.66Nolomirole HCl
CAS:Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFórmula:C19H28ClNO4Pureza:100% - 99.12%Forma y color:SolidPeso molecular:369.88Brexpiprazole S-oxide
CAS:Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Fórmula:C25H27N3O3SPureza:98%Forma y color:SolidPeso molecular:449.57Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Fórmula:C18H21NSPureza:100% - 98.58%Forma y color:SolidPeso molecular:283.43UNC10099984A
CAS:UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a Ki value of 4.6 nM and an EC50 of 6.2 nM for β-arrestin. This compound is useful for research into central nervous system diseases related to the D2 receptor.Fórmula:C24H29Cl2N3O2Forma y color:SolidPeso molecular:462.41Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Fórmula:C24H23ClF3NPureza:99.99%Forma y color:SolidPeso molecular:417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Fórmula:C19H19NSPureza:97.50%Forma y color:SolidPeso molecular:293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Methyldopa hydrate
CAS:Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Fórmula:C10H13NO4H2OPureza:99.67%Forma y color:White SolidPeso molecular:238.24Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.Fórmula:C23H27F3N2O3Pureza:98.10%Forma y color:SoildPeso molecular:436.47L-DOPA
CAS:L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Fórmula:C9H11NO4Pureza:98.99% - 99.93%Forma y color:Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidPeso molecular:197.19Abaperidone
CAS:Abaperidone is an atypical antipsychotic, antagonizes 5-HT2A (IC50=6.2 nM) and D2 receptors (IC50=17 nM), reduces hsp70 mRNA in rat brains.Fórmula:C25H25FN2O5Pureza:94.35%Forma y color:SolidPeso molecular:452.47A-77636
CAS:A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Fórmula:C20H27NO3Pureza:98%Forma y color:SolidPeso molecular:329.43Diclofensine
CAS:Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Fórmula:C17H17Cl2NOPureza:98.08%Forma y color:SolidPeso molecular:322.23Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Fórmula:C21H26ClNPureza:99.99%Forma y color:Crystalline SolidPeso molecular:327.9Ref: TM-T4274
10mg47,00€25mg67,00€50mg87,00€100mg116,00€200mg170,00€500mg279,00€1mL*10mM (DMSO)50,00€BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Fórmula:C26H31N3O2Pureza:99.44%Forma y color:SolidPeso molecular:417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Fórmula:C21H25NO4Pureza:100% - 99.8%Forma y color:Off-White SolidPeso molecular:355.43Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Fórmula:C24H27FN2O4Pureza:99.42%Forma y color:SolidPeso molecular:426.48D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Fórmula:C27H37NO5Pureza:98%Forma y color:SolidPeso molecular:455.59Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFórmula:C10H13NO4Pureza:99.86% - 99.89%Forma y color:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Fórmula:C28H36N4O2S·HClPureza:99.51%Forma y color:SolidPeso molecular:529.14
