
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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Ergocornine
CAS:Ergocornine is a naturally occurring ergot alkaloid and acts as a dopamine receptor (dopamine receptor) agonist.Fórmula:C31H39N5O5Forma y color:SolidPeso molecular:561.67Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Atomoxetine hydrochloride
CAS:Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Fórmula:C17H22ClNOPureza:99.86%Forma y color:White SolidPeso molecular:291.82Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Forma y color:Almost White To White Crystalline PowderPeso molecular:351.935-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Fórmula:C18H20N2OPureza:96.33%Forma y color:SolidPeso molecular:280.36Ropinirole hydrochloride
CAS:Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Fórmula:C16H24N2O·HClPureza:99.87% - 99.98%Forma y color:Off-White SolidPeso molecular:296.84UCSF924
CAS:UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Fórmula:C20H22N2O2Pureza:98%Forma y color:SolidPeso molecular:322.4Medifoxamine
CAS:Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFórmula:C16H19NO2Pureza:98.35%Forma y color:SolidPeso molecular:257.33Ref: TM-T24444
1mg99,00€5mg235,00€10mg354,00€25mg635,00€50mg893,00€100mg1.159,00€1mL*10mM (DMSO)259,00€DOPEXAMINE
CAS:Dopexamine is a dopaminergic agonistFórmula:C22H32N2O2Pureza:99.42%Forma y color:SolidPeso molecular:356.5Ref: TM-T8653
1mg131,00€2mg188,00€5mg284,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)306,00€Trimipramine maleate
CAS:Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Fórmula:C24H30N2O4Pureza:99.47%Forma y color:SolidPeso molecular:410.51Dopamine D2 receptor agonist-2
CAS:Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.Fórmula:C25H31Cl2N5OSPureza:98.93%Forma y color:SoildPeso molecular:520.52Ref: TM-T60075
1mg38,00€5mg71,00€10mg90,00€25mg148,00€50mg210,00€100mg314,00€200mg452,00€1mL*10mM (DMSO)90,00€Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Fórmula:C20H25ClN2OSPureza:99.17%Forma y color:SolidPeso molecular:376.94Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.45% - 99.89%Forma y color:SolidPeso molecular:477.57Fluphenazine dihydrochloride
CAS:Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Fórmula:C22H28Cl2F3N3OSPureza:99.23%Forma y color:Off-White SolidPeso molecular:510.44Thiethylperazine dimaleate
CAS:Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.Fórmula:C30H37N3O8S2Pureza:99.07%Forma y color:SolidPeso molecular:631.76carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.Fórmula:C24H31N3O2SPureza:98.15%Forma y color:SolidPeso molecular:425.59Trifluoperazine
CAS:Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Fórmula:C21H24F3N3SPureza:98.3% - 99.46%Forma y color:White To Yellowish Crystalline PowderPeso molecular:407.5(-)-GSK598809 hydrochloride
CAS:(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.Fórmula:C22H24ClF4N5OSPureza:97.66%Forma y color:SoildPeso molecular:517.97Molindone
CAS:Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.Fórmula:C16H24N2O2Pureza:98% - 99.37%Forma y color:Off-White SolidPeso molecular:276.37Foscarbidopa
CAS:Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Fórmula:C10H15N2O7PPureza:98%Forma y color:SolidPeso molecular:306.21