CymitQuimica logo
Src

Src

Os inibidores de Src são compostos que têm como alvo as quinases da família Src, que estão envolvidas em vários processos celulares, incluindo crescimento, diferenciação e angiogênese. As quinases Src desempenham um papel crucial nas vias de sinalização que promovem a formação de novos vasos sanguíneos em tumores. Ao inibir Src, é possível interromper essas vias, reduzindo assim a angiogênese e o crescimento tumoral. Os inibidores de Src são amplamente utilizados na pesquisa do câncer e no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma seleção abrangente de inibidores de Src de alta qualidade para apoiar sua pesquisa em oncologia, sinalização celular e angiogênese.

Produtos da "Src"

Ordenar por

produtos por página.82 produtos desta categoria.
  • Tolimidone

    CAS:
    Tolimidone (NSC 314335) is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.
    Fórmula:C11H10N2O2
    Pureza:99.85% - 99.85%
    Cor e Forma:Solid
    Peso molecular:202.21

    Ref: TM-T6896

    5mg
    50,00€
    10mg
    77,00€
    25mg
    117,00€
    50mg
    180,00€
    100mg
    270,00€
    1mL*10mM (DMSO)
    52,00€
  • WHI-P154

    CAS:
    Fórmula:C16H14BrN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:376.2047

    Ref: IN-DA00BF57

    1g
    597,00€
    10mg
    68,00€
    50mg
    118,00€
    100mg
    187,00€
    250mg
    224,00€
  • TL02-59 dihydrochloride

    CAS:
    TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).
    Fórmula:C32H36Cl2F3N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:682.56

    Ref: TM-T13186L

    10mg
    A consultar
    50mg
    A consultar
  • A-770041

    CAS:
    A-770041 is an Lck inhibitor, YZ inhibits the production of IL-2 stimulated by concanavalin A in whole blood, and can prevent cardiac allograft rejection.
    Fórmula:C34H39N9O3
    Pureza:99.23% - 99.86%
    Cor e Forma:Solid
    Peso molecular:621.73

    Ref: TM-T14074

    1mg
    55,00€
    5mg
    116,00€
    10mg
    188,00€
    25mg
    426,00€
    50mg
    725,00€
    100mg
    1.130,00€
    200mg
    1.501,00€
    1mL*10mM (DMSO)
    159,00€
  • A 419259 trihydrochloride

    CAS:
    A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, 3 nM and 3 nM for Src, Lck and Lyn).
    Fórmula:C29H37Cl3N6O
    Pureza:100% - 99.47%
    Cor e Forma:Solid
    Peso molecular:592

    Ref: TM-TQ0132

    1mg
    52,00€
    2mg
    74,00€
    5mg
    107,00€
    10mg
    170,00€
    25mg
    319,00€
    50mg
    557,00€
    100mg
    797,00€
    500mg
    1.586,00€
  • GluR6 antagonist-1

    CAS:
    GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.
    Fórmula:C15H11ClN2OS
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:302.78

    Ref: TM-T9723

    2mg
    38,00€
    5mg
    58,00€
    10mg
    90,00€
    25mg
    138,00€
    50mg
    197,00€
    100mg
    294,00€
    200mg
    411,00€
    1mL*10mM (DMSO)
    65,00€
  • KX1-004

    CAS:
    KX1-004, a potential protective drug for NIHL, is an effective small molecule inhibitor of Src-PTK.
    Fórmula:C16H13FN2O2
    Pureza:99.12% - ≥95%
    Cor e Forma:Solid
    Peso molecular:284.29

    Ref: TM-T1812

    1mg
    46,00€
    2mg
    59,00€
    5mg
    87,00€
    10mg
    160,00€
    25mg
    283,00€
    50mg
    465,00€
    100mg
    655,00€
    500mg
    1.378,00€
    1mL*10mM (DMSO)
    97,00€
  • Dasatinib monohydrate

    CAS:
    Dasatinib monohydrate, an oral SRC-kinase inhibitor, counters imatinib-resistant chronic myeloid leukemia.
    Fórmula:C22H28ClN7O3S
    Pureza:100% - 99.68%
    Cor e Forma:Solid
    Peso molecular:506.03

    Ref: TM-T1448L

    50mg
    39,00€
    100mg
    55,00€
    200mg
    72,00€
    500mg
    104,00€
    1mL*10mM (DMSO)
    48,00€
  • Src Inhibitor 1

    CAS:
    Src Inhibitor 1 (Src Kinase Inhibitor 1) is a potent and selective dual site Src tyrosine kinase inhibitor.
    Fórmula:C22H19N3O3
    Pureza:100% - 99.38%
    Cor e Forma:Solid
    Peso molecular:373.4

    Ref: TM-T3593

    1mg
    39,00€
    2mg
    52,00€
    5mg
    73,00€
    10mg
    90,00€
    25mg
    207,00€
    50mg
    373,00€
    100mg
    547,00€
    500mg
    1.159,00€
  • MCB-613

    CAS:
    MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.
    Fórmula:C20H20N2O
    Pureza:98.17% - 99.33%
    Cor e Forma:Solid
    Peso molecular:304.39

    Ref: TM-T6886

    1mg
    46,00€
    2mg
    59,00€
    5mg
    87,00€
    10mg
    144,00€
    25mg
    259,00€
    50mg
    378,00€
    100mg
    567,00€
    1mL*10mM (DMSO)
    96,00€
  • 1-Naphthyl PP1 hydrochloride

    CAS:
    1-Naphthyl PP1 hydrochloride (1-NA-PP 1 hydrochloride) is a selective inhibitor of src family kinases v-Src
    Fórmula:C19H20ClN5
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:353.85

    Ref: TM-T7371

    5mg
    46,00€
    10mg
    65,00€
    25mg
    123,00€
    50mg
    192,00€
    100mg
    298,00€
    200mg
    430,00€
    1mL*10mM (DMSO)
    49,00€
  • NVP-BHG 712

    CAS:
    Fórmula:C26H20F3N7O
    Pureza:>95.0%(HPLC)
    Cor e Forma:White to Light yellow to Light orange powder to crystal
    Peso molecular:503.49

    Ref: 3B-N1099

    10mg
    128,00€
    50mg
    426,00€
  • SI-2 hydrochloride

    CAS:
    SI-2 hydrochloride, an SRC-3 inhibitor, induces breast cancer cell death (IC50: 3-20 nM) with good oral bioavailability.
    Fórmula:C15H16ClN5
    Pureza:98.18%
    Cor e Forma:Solid
    Peso molecular:301.77

    Ref: TM-T12906

    5mg
    35,00€
    10mg
    47,00€
    25mg
    64,00€
    50mg
    A consultar
  • 1-NM-PP1

    CAS:
    1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
    Fórmula:C20H21N5
    Pureza:98% - 98.93%
    Cor e Forma:White Cyrstalline Solid
    Peso molecular:331.41

    Ref: TM-T2153

    1mg
    50,00€
    2mg
    66,00€
    5mg
    88,00€
    10mg
    139,00€
    25mg
    286,00€
    50mg
    532,00€
    100mg
    705,00€
    1mL*10mM (DMSO)
    95,00€
  • Rebastinib

    CAS:
    DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,
    Fórmula:C30H28FN7O3
    Pureza:99.53% - 99.79%
    Cor e Forma:Solid
    Peso molecular:553.59

    Ref: TM-T2640

    2mg
    48,00€
    5mg
    69,00€
    10mg
    96,00€
    25mg
    172,00€
    50mg
    251,00€
    100mg
    378,00€
    200mg
    567,00€
  • PP 2

    CAS:
    Fórmula:C15H16ClN5
    Pureza:>97.0%(T)(HPLC)
    Cor e Forma:White to Light yellow powder to crystal
    Peso molecular:301.78

    Ref: 3B-P2833

    10mg
    142,00€
    50mg
    462,00€
  • AMG-47a

    CAS:
    AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.
    Fórmula:C29H28F3N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:535.56

    Ref: TM-T7123

    1mg
    46,00€
    5mg
    87,00€
    10mg
    153,00€
    25mg
    249,00€
    50mg
    369,00€
    100mg
    545,00€
    1mL*10mM (DMSO)
    96,00€
  • Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Fórmula:C9H11NO3·HCl
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:217.65

    Ref: TM-T0948

    1g
    145,00€
    50mg
    35,00€
    100mg
    50,00€
    500mg
    97,00€
  • Pyridostatin

    CAS:
    Pyridostatin (RR82) is a synthetic small-molecule stabilizer of G-quadruplexes, a secondary structure of DNA that usually exists in the end of the chromosome or
    Fórmula:C31H32N8O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:596.64

    Ref: TM-T1899

    1mg
    42,00€
    5mg
    81,00€
    10mg
    111,00€
    25mg
    190,00€
    50mg
    298,00€
    1mL*10mM (DMSO)
    115,00€
  • PP2

    CAS:
    PP2 (AG 1879,AGL 1879) is a effective inhibitor of Lck/Fyn (IC50:4/5 nM) , ~100-fold less potent to EGFR, inactive for ZAP-70, PKA and JAK2.
    Fórmula:C15H16ClN5
    Pureza:95.65% - 98%
    Cor e Forma:White Solid
    Peso molecular:301.77

    Ref: TM-T6266

    2mg
    47,00€
    5mg
    69,00€
    10mg
    116,00€
    25mg
    188,00€
    50mg
    321,00€
    100mg
    510,00€
    200mg
    725,00€
    1mL*10mM (DMSO)
    74,00€