Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
Sort by
LSD1-UM-109
CAS:LSD1-UM-109 is a highly potent and reversible inhibitor of LSD1, demonstrating an IC50 of 3.1 nM.Formula:C29H27FN6Purity:98%Color and Shape:SolidMolecular weight:478.56JAK-IN-5
CAS:JAK-IN-5 is a JAK inhibitor.Formula:C27H31FN6OPurity:97.78% - 98.78%Color and Shape:SolidMolecular weight:474.57Ref: TM-T11710
1mg187.00€5mg391.00€10mg582.00€25mg929.00€50mg1,254.00€100mg1,691.00€500mg3,382.00€1mL*10mM (DMSO)567.00€PARP7-IN-15
CAS:PARP7-IN-15 (Compound 18) is a potent PARP7 inhibitor exhibiting an IC50 of 0.56 nM and demonstrates antitumor activity [1].Formula:C23H24F6N6O4Purity:98%Color and Shape:SolidMolecular weight:562.46Pulrodemstat
CAS:Pulrodemstat (CC-90011) is an LSD1 inhibitor with anticancer and antitumor activity, inhibiting proliferation and migration of HNSCC cells.Formula:C24H23F2N5O2Purity:98.11% - 98.89%Color and Shape:SolidMolecular weight:451.47KF21213
CAS:KF21213 shows a high affinity for the adenosine A2A receptors (Ki=3.0 nM). KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors.Formula:C19H22N4O3Purity:98%Color and Shape:SolidMolecular weight:354.4Pim-1 kinase inhibitor 8
CAS:Pim-1 kinase inhibitor 8 is a Pim-1 kinase inhibitor with anticancer activity that inhibits cell migration and can be studied in breast cancer.Formula:C14H17N3O3Purity:99.81%Color and Shape:SoildMolecular weight:275.3Menin-MLL inhibitor 20
CAS:Menin-MLL inhibitor 20 is an irreversible inhibitor of menin-MLL interaction with antitumor activities.Formula:C33H40N8O4Purity:98.89%Color and Shape:SolidMolecular weight:612.72Ref: TM-T9399
1mg40.00€5mg90.00€10mg135.00€25mg264.00€50mg390.00€100mg555.00€200mg752.00€1mL*10mM (DMSO)90.00€KSQ-4279
CAS:KSQ-4279 (USP1-IN-1) is an inhibitor of USP1 and PARP.KSQ-4279 has anticancer activity and is used in the study of non-small cell lung cancer, osteosarcoma,Formula:C27H25F3N8OPurity:99.43% - 99.76%Color and Shape:SoildMolecular weight:534.54CCT129202
CAS:CCT129202 is an ATP-competitive pan-Aurora inhibitor for Aurora A, Aurora B and Aurora C with IC50 of 0.042 μM, 0.198 μM and 0.227 μM, respectively.Formula:C23H25ClN8OSPurity:98.14%Color and Shape:SolidMolecular weight:497.025-Hydroxymethyl-2'-deoxycytidine
CAS:5-Hydroxymethyl-2'-deoxycytidine is an oxidized derivative of 5-methyl-2'-deoxycytidine (5-mdC) in DNA, causing DNA damage reactions, chromosomal aberrations,Formula:C10H15N3O5Purity:99.8%Color and Shape:SolidMolecular weight:257.24Ref: TM-T40834
1mg40.00€5mg88.00€10mg119.00€25mg202.00€50mg323.00€100mg487.00€500mg1,035.00€1mL*10mM (DMSO)87.00€Uzansertib phosphate
CAS:Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, PIM2 and PIM3.Formula:C26H29F3N5O7PPurity:99.75% - 99.85%Color and Shape:SolidMolecular weight:611.51MI-503
CAS:MI-503 is an efficient and selective Menin-MLL inhibitor. MI-503 has a significant inhibitory effect on human MLL leukemia cell line. Cost-effective and quality-assured.Formula:C28H27F3N8SPurity:99.87% - 99.99%Color and Shape:SolidMolecular weight:564.63Ref: TM-TQ0069
2mg115.00€5mg208.00€10mg348.00€25mg520.00€50mg750.00€100mg1,035.00€200mg1,406.00€1mL*10mM (DMSO)259.00€BRD7-IN-3
BRD7-IN-3 (compound 1-78) functions as a dual inhibitor targeting the bromodomain-containing proteins BRD7 and BRD9, demonstrating half-maximal inhibitoryFormula:C18H18N2O2Purity:98%Color and Shape:SolidMolecular weight:294.35JPHM-2-167
CAS:PHM-2-167 (Compound 11) is a selective inhibitor of the prolyl hydroxylase domain enzyme (PHD). It inhibits PHD2 and PHD3 with IC50 values of 0.253 μM and 3.95 μM, respectively. PHM-2-167 is applicable for research in chronic kidney disease.Formula:C30H28N6O2Color and Shape:SolidMolecular weight:504.582GSK2807 Trifluoroacetate
CAS:GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM).Formula:C21H33F3N8O7Purity:99.95%Color and Shape:SolidMolecular weight:566.53CARM1-IN-1
CAS:CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM.Formula:C26H21Br2NO3Purity:97.35%Color and Shape:SolidMolecular weight:555.26Ref: TM-T10682L
1mg37.00€5mg88.00€10mg127.00€25mg250.00€50mg406.00€100mg632.00€200mg883.00€1mL*10mM (DMSO)97.00€Golidocitinib
CAS:Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, >30 μM).Formula:C25H31N9O2Purity:100% - 98.87%Color and Shape:SolidMolecular weight:489.57Ref: TM-T10431
2mg96.00€5mg163.00€10mg268.00€25mg465.00€50mg618.00€100mg880.00€1mL*10mM (DMSO)170.00€AZD-2461
CAS:AZD2461 is a novel PARP inhibitor.Formula:C22H22FN3O3Purity:98% - 99.25%Color and Shape:SolidMolecular weight:395.43PRMT5-IN-2
CAS:PRMT5-IN-2 is an inhibitor of protein arginine methyltransferase 5.Formula:C17H16ClFN4O4Purity:98%Color and Shape:SolidMolecular weight:394.78JI069
CAS:JI069 (WAY-354189) is a potent STAT3 inhibitor that inhibits gp130 signaling by inducing dissociation between gp130 and JAK1.Formula:C15H12Cl2N2O4SPurity:98.01%Color and Shape:SolidMolecular weight:387.24
