Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
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SETDB1-TTD-IN-1
CAS:SETDB1-TTD-IN-1 is a potent and selective inhibitor of SET domain bifurcated protein 1 tandem tudor domain (SETDB1-TTD, Kd = 88 nM).Cost-effective and quality-assured.Formula:C28H31N5O2Purity:98.26% - 99.38%Color and Shape:SolidMolecular weight:469.58MRS2698
CAS:MRS2698: potent P2Y2 agonist, EC50 8 nM, >300x selectivity over P2Y4/P2Y6.Formula:C9H16N3O13P3SPurity:98%Color and Shape:SolidMolecular weight:499.22Dot1L-IN-1
CAS:The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.Formula:C32H36ClN9O2SPurity:98%Color and Shape:SolidMolecular weight:646.21Ryuvidine
CAS:Ryuvidine is a dual inhibitor of KDM5A and SETD8, an inducer of the DNA damage response, and can be used to study breast cancer and erythroderma.Formula:C15H12N2O2SPurity:98.6%Color and Shape:SolidMolecular weight:284.33Menin-MLL inhibitor 27
Menin-MLL inhibitor 27 effectively inhibits the interaction between Menin and MLL, serving as a potential tool in cancer research, particularly for acuteFormula:C31H35FN8O2Purity:98%Color and Shape:SolidMolecular weight:570.66ZL0420
CAS:ZL0420: Potent, selective BRD4 inhibitor, IC50 27 nM BD1 & 32 nM BD2.Formula:C16H16N4O2Purity:97.77%Color and Shape:SolidMolecular weight:296.32Ref: TM-T6828
2mg42.00€5mg64.00€10mg101.00€25mg197.00€50mg340.00€100mg484.00€200mg645.00€1mL*10mM (DMSO)70.00€Iadademstat dihydrochloride
CAS:Iadademstat dihydrochloride (ORY-1001(trans)) , a Potent and Selective Covalent KDM1A/LSD1 Inhibitor, for the Treatment of Acute Leukemia.Formula:C15H24Cl2N2Purity:99.78%Color and Shape:SolidMolecular weight:303.27PIM1-IN-1
CAS:PIM1-IN-1 inhibits PIM1/3 with IC50s: PIM1 (7 nM), PIM2 (5530 nM), PIM3 (70 nM); it has anti-cancer properties.Formula:C25H30N8O2Purity:98%Color and Shape:SolidMolecular weight:474.56BMS-986158
CAS:BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.Formula:C30H33N5O2Purity:98.78%Color and Shape:SolidMolecular weight:495.62Ref: TM-T14685
1mg87.00€5mg259.00€10mg465.00€25mg745.00€50mg1,026.00€100mg1,388.00€1mL*10mM (DMSO)283.00€GNE-207
CAS:GNE-207 is a selective and orally bioavailable inhibitor of the bromodomain of CBP (IC50: 1 nM).Formula:C29H30N6O3Purity:98%Color and Shape:SolidMolecular weight:510.59HIF-2α-IN-2
CAS:HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).Formula:C17H13F2NO4SPurity:99.24%Color and Shape:SolidMolecular weight:365.35Ref: TM-T11561
1mg71.00€5mg135.00€10mg178.00€25mg309.00€50mg447.00€100mg620.00€200mg835.00€1mL*10mM (DMSO)149.00€A1874
CAS:A1874 is a nutlin-based and BRD4-degrading PROTAC which induces BRD4 degradation in cells. Effective in inhibiting many cancer cell lines proliferation.Formula:C58H62Cl3F2N9O7SPurity:99.52%Color and Shape:SolidMolecular weight:1173.59TP-472
CAS:TP-472 is a selective inhibitor of BRD9 (Kd: 33 nM).Formula:C20H19N3O2Purity:98%Color and Shape:SolidMolecular weight:333.38JDTic dihydrochloride
CAS:JDTic is a powerful antagonist of kappa-opioid receptors (KOR), effectively inhibiting the antinociceptive effects induced by the κ-agonist U50, 488.Formula:C28H41Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:538.55PARP/PI3K-IN-1
CAS:PARP/PI3K-IN-1 is a PARP and PI3K dual inhibitor with anticancer and antiproliferative activities for the study of breast, pancreatic and lung cancers.Formula:C33H28F4N8O3Purity:99.59%Color and Shape:SolidMolecular weight:660.62HS94
CAS:HS94 (DAPK3 inhibitor HS94) is a selective and potent DAPK3 inhibitor with a Ki value of 126 nM for Pim kinase inhibition and can be used to study hypertension.Formula:C15H15N5O2SPurity:95.04%Color and Shape:SolidMolecular weight:329.382-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
CAS:2-methyl-2,3-dihydro-1,5-benzothiazepin-4(5H)-one is ligand of CBP.Formula:C10H11NOSPurity:99.68%Color and Shape:SolidMolecular weight:193.27ABBV-744
CAS:ABBV-744 is a BDII-selective BET bromodomain inhibitor that inhibits BRD2/3/4. It is used in the research on inflammatory diseases, cancer, and AIDS.Formula:C28H30FN3O4Purity:100% - 99.79%Color and Shape:SolidMolecular weight:491.55Ref: TM-T4697
1mg47.00€2mg59.00€5mg96.00€10mg150.00€25mg299.00€50mg432.00€100mg527.00€200mg758.00€1mL*10mM (DMSO)96.00€Butyrolactone 3
CAS:Butyrolactone 3 (MB-3) is a Gcn5 inhibitor with weak affinity for CBP.Butyrolactone 3 has antimicrobial activity and can be used in cancer.Formula:C9H12O4Purity:98.99% - 99.5%Color and Shape:SolidMolecular weight:184.19Menin-MLL inhibitor 29
Menin-MLL Inhibitor 29 (Compound C1) is a Menin-MLL protein-protein interaction (PPI) inhibitor that demonstrates high affinity to Menin with a dissociationFormula:C36H26Br2F6N4PRhPurity:98%Color and Shape:SolidMolecular weight:922.3
