Phospholipase
Phospholipases are a group of enzymes that hydrolyze phospholipids into fatty acids and other lipophilic substances, playing a critical role in membrane biology and the generation of signaling molecules. Inhibitors of phospholipases are used to study their role in inflammatory diseases, cardiovascular disorders, and neurodegeneration. These inhibitors are also valuable in exploring lipid signaling pathways and their implications in disease mechanisms. At CymitQuimica, we provide a variety of phospholipase inhibitors to support your research in inflammation, lipid metabolism, and cell signaling.
Products of "Phospholipase"
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hnps-PLA Inhibitor
CAS:Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).Formula:C21H21N3O4Purity:98.95%Color and Shape:SolidMolecular weight:379.41Ref: TM-T4192
1mg56.00€2mg81.00€5mg119.00€10mg202.00€25mg341.00€50mg509.00€100mg725.00€1mL*10mM (DMSO)137.00€RHC 80267
CAS:RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Formula:C20H34N4O4Purity:99.54%Color and Shape:White SolidMolecular weight:394.51Compound 48/80 trihydrochloride
CAS:Compound 48/80 trihydrochloride (C48/80 trihydrochloride) 是 N-甲基对甲氧基苯乙胺和甲醛发生缩合反应后的混合物。Compound 48/80 trihydrochloride 是一种肥大细胞 (mast cell) 脱颗粒剂和组胺 (histamine) 释放剂。Compound 48/80 trihydrochloride 对人血小板磷脂酰肌醇特异性磷脂酶 C (phosphatidylinositol-specific phospholipase C) 活性有抑制作用。Formula:C32H48Cl3N3O3Purity:98%Color and Shape:SolidMolecular weight:629.1Rilapladib
CAS:Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormula:C40H38F5N3O3SPurity:97.29%Color and Shape:SolidMolecular weight:735.8Ref: TM-T16751
1mg93.00€5mg227.00€10mg369.00€25mg622.00€50mg885.00€100mg1,206.00€1mL*10mM (DMSO)369.00€CAY10594
CAS:CAY10594, a PLD2 inhibitor, mitigates acetaminophen liver damage via the p-GSK-3β/JNK pathway.Formula:C26H28N4O2Purity:98%Color and Shape:SolidMolecular weight:428.53Melittin
CAS:Melittin: principal bee venom toxin, 26 amino acids, activates low-weight PLA2, not high-weight PLA2.Formula:C131H229N39O31Purity:98.37% - 99.14%Color and Shape:SolidMolecular weight:2846.46RPI-1
CAS:RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.Formula:C17H15NO4Purity:98.28% - ≥95%Color and Shape:SolidMolecular weight:297.31DPTIP
CAS:DPTIP is an effective inhibitor of neutral sphingomyelinase 2 with an IC50 value of 30 nM.Formula:C21H18N2O3SPurity:98.80%Color and Shape:SolidMolecular weight:378.44Ref: TM-T60043
1mg48.00€2mg63.00€5mg96.00€10mg153.00€25mg298.00€50mg487.00€100mg710.00€1mL*10mM (DMSO)96.00€5-HT1A modulator 1
CAS:5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formula:C21H25N3O2SPurity:99.66%Color and Shape:SolidMolecular weight:383.51(E/Z)-Polydatin
CAS:(E/Z)-Polydatin, a resveratrol glycoside from Picea/Polygonum, in grapes & chocolate, has anti-inflammatory and anti-cancer properties.Formula:C20H22O8Purity:98.78% - 99.16%Color and Shape:SolidMolecular weight:390.38Darapladib
CAS:Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.Formula:C36H38F4N4O2SPurity:100% - 99.82%Color and Shape:SolidMolecular weight:666.77Ref: TM-T6109
1mg52.00€2mg70.00€5mg96.00€10mg169.00€25mg329.00€50mg535.00€100mg747.00€500mg1,510.00€1mL*10mM (DMSO)154.00€ASM-IN-3
CAS:ASM-IN-3 (Compound 21b) is a selective acid sphingomyelinase (ASM) inhibitor that can penetrate the blood-brain barrier, with an IC50 of 3.37 μM against purified human ASM. By inhibiting ASM activity in the hippocampus and promoting neurogenesis, ASM-IN-3 alleviates depressive-like behavior in reserpine-induced depressive rats.Formula:C17H13ClN2O4Color and Shape:SolidMolecular weight:344.75Desketoraloxifene
CAS:Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).Formula:C27H27NO3SPurity:98%Color and Shape:SolidMolecular weight:445.57Bromoenol lactone
CAS:NeurokininBromoenol lactone ((6E)-Bromoenol lactone) is an iPLA2β and serine protease inhibitor that attenuates nicotine-induced breast cancer cell proliferation.Formula:C16H13BrO2Color and Shape:SolidMolecular weight:317.18Tanshinone I
CAS:Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.Formula:C18H12O3Purity:98.31% - 98.70%Color and Shape:SolidMolecular weight:276.291-Naphthaleneacetic acid potassium salt
CAS:1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.Formula:C12H9O2·KPurity:97.68%Color and Shape:Off-White To Beige PowderMolecular weight:224.3ML-095 hydrochloride
CAS:ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.Formula:C13H15ClN2O3Purity:98.18%Color and Shape:SolidMolecular weight:282.72Ref: TM-T21969
2mg38.00€5mg58.00€10mg96.00€25mg170.00€50mg298.00€100mg432.00€200mg607.00€1mL*10mM (DMSO)64.00€Halobetasol propionate
CAS:Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.Formula:C25H31ClF2O5Purity:99.89%Color and Shape:Distributed As 0 05% OintmentMolecular weight:484.96AA26-9
CAS:AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Formula:C7H10N4OPurity:99.88%Color and Shape:SolidMolecular weight:166.18Ref: TM-T3990
1mg37.00€2mg52.00€5mg79.00€10mg119.00€25mg210.00€50mg350.00€100mg522.00€1mL*10mM (DMSO)87.00€VU533
CAS:VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.Formula:C21H22FN3O3S2Purity:99.08%Color and Shape:SolidMolecular weight:447.55
