AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurity:99.76%Color and Shape:White PowderMolecular weight:473.39Ref: TM-T16126
1mg87.00€5mg250.00€10mg359.00€25mg707.00€50mg1,017.00€100mg1,454.00€1mL*10mM (DMSO)274.00€Benzethonium chloride
CAS:Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.Formula:C27H42ClNO2Purity:99.91%Color and Shape:White To Off-White Solid Solid Particulate/PowderMolecular weight:448.09(Rac)-Sabcomeline HCl
CAS:Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.Formula:C10H16ClN3OPurity:99.03%Color and Shape:SoildMolecular weight:229.71Mivacurium dichloride
CAS:Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.Formula:C58H80Cl2N2O14Purity:99.2% - 99.48%Color and Shape:Off-White SolidMolecular weight:1100.17Ref: TM-T22371
2mg48.00€5mg69.00€10mg89.00€25mg130.00€50mg198.00€100mg303.00€200mg457.00€1mL*10mM (DMSO)96.00€(S)-(+)-Dimethindene maleate
CAS:(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormula:C24H28N2O4Purity:99.43%Color and Shape:SolidMolecular weight:408.49Benactyzine hydrochloride
CAS:Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.Formula:C20H26ClNO3Purity:100% - 99.68%Color and Shape:SolidMolecular weight:363.88Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Formula:C11H16N2OPurity:98%Color and Shape:SolidMolecular weight:192.26CP-810123
CAS:CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.Formula:C14H18N4OPurity:98.63% - 99.23%Color and Shape:SolidMolecular weight:258.32Pozanicline hydrochloride
Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.Formula:C11H17ClN2OPurity:99.6%Color and Shape:SolidMolecular weight:228.72Ref: TM-T16563L
1mg77.00€5mg155.00€10mg220.00€25mg338.00€50mg472.00€100mg632.00€200mg853.00€1mL*10mM (DMSO)134.00€Gallamine triethiodide
CAS:Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.Formula:C30H60I3N3O3Purity:98.90%Color and Shape:White Amorphous Powder SolidMolecular weight:891.53Donepezil Hydrochloride
CAS:Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).Formula:C24H29NO3·HClPurity:99.55% - 99.8%Color and Shape:White To Off-White Crystalline SolidMolecular weight:415.969-CP-Ade Mesylate
CAS:9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.Formula:C11H17N5O3SPurity:99.91%Color and Shape:SolidMolecular weight:299.35PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Formula:C15H17N3O2Purity:99% - 99.48%Color and Shape:SolidMolecular weight:271.31Ref: TM-T23145
1mg50.00€5mg107.00€10mg170.00€25mg378.00€50mg645.00€100mg945.00€500mg2,052.00€1mL*10mM (DMSO)105.00€Afacifenacin
CAS:Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.Formula:C27H26F3N3O2Purity:99.57%Color and Shape:SolidMolecular weight:481.51(-)-OPC-51803
CAS:(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.Formula:C26H32ClN3O2Purity:100% - 100.00%Color and Shape:SoildMolecular weight:454NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.Formula:C14H8N4OPurity:98.81%Color and Shape:SolidMolecular weight:248.24Ref: TM-T28199
1mg46.00€5mg96.00€10mg144.00€25mg298.00€50mg469.00€100mg687.00€500mg1,444.00€1mL*10mM (DMSO)97.00€TMPH
CAS:TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.Formula:C16H31NO2Purity:99.78%Color and Shape:SoildMolecular weight:269.42Ref: TM-T60080
2mg38.00€5mg58.00€10mg88.00€25mg140.00€50mg215.00€100mg319.00€200mg449.00€1mL*10mM (DMSO)57.00€DL-trihexyphenidyl hydrochloride
CAS:DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.Formula:C20H32ClNOPurity:99.63% - 99.71%Color and Shape:SolidMolecular weight:337.93(S)-UFR2709 hydrochloride
CAS:(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in rats, studies nicotine addiction.Formula:C13H18ClNO2Purity:98.94%Color and Shape:SolidMolecular weight:255.74Ref: TM-T37094
1mg42.00€5mg88.00€10mg120.00€25mg235.00€50mg354.00€100mg550.00€500mg1,159.00€1mL*10mM (DMSO)92.00€Acetamiprid
CAS:Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.Formula:C10H11ClN4Purity:99.66%Color and Shape:White PowderMolecular weight:222.67
