Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Fórmula:C19H21NPureza:99.05% - 99.23%Forma y color:SolidPeso molecular:263.38YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Fórmula:C14H17N3OPureza:98%Forma y color:SolidPeso molecular:243.38-OH-Dpat
CAS:8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Fórmula:C16H25NOPureza:98%Forma y color:SolidPeso molecular:247.38Ethylpropyltryptamine
CAS:Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Fórmula:C15H22N2Forma y color:SolidPeso molecular:230.35Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Fórmula:C24H32ClNO6Pureza:99.73%Forma y color:Colorless LiquidPeso molecular:465.97Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFórmula:C20H24N2O6SPureza:100%Forma y color:White PowderPeso molecular:420.48Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOForma y color:SolidPeso molecular:301.47NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H25N3O2SPureza:98%Forma y color:SolidPeso molecular:431.55AAZ-A 154 benzoate
CAS:AAZ-A 154 benzoate is a selective, competitive, and non-hallucinogenic 5-HT2AR antagonist. This compound facilitates neuronal growth in rodents and produces lasting beneficial behavioral effects.Fórmula:C21H26N2O3Forma y color:SolidPeso molecular:354.44Nardosinonediol
CAS:Nardosinonediol is a natural compound derived from Nardostachys jatamansi that acts as a SERT inhibitor, regulating serotonin levels and antidepressant.Fórmula:C15H24O3Pureza:98%Forma y color:SolidPeso molecular:252.35Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Fórmula:C19H19NSPureza:97.50%Forma y color:SolidPeso molecular:293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€SB-269970 hydrochloride
CAS:SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFórmula:C18H28N2O3S·HClPureza:98.45%Forma y color:SolidPeso molecular:388.95Ogerin
CAS:Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Fórmula:C17H17N5OPureza:99.50% - 99.75%Forma y color:SolidPeso molecular:307.35Ref: TM-T16378
1mg35,00€2mg52,00€5mg74,00€10mg115,00€25mg227,00€50mg380,00€100mg567,00€1mL*10mM (DMSO)86,00€Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.83%Forma y color:SolidPeso molecular:575.61Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Fórmula:C21H24N2Pureza:99.76%Forma y color:SolidPeso molecular:304.43PF-03382792
CAS:PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Fórmula:C23H32FN3O4Pureza:98.09%Forma y color:SolidPeso molecular:433.52NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Fórmula:C25H26ClN3O2SPureza:99.8%Forma y color:SoildPeso molecular:468.01Ref: TM-T12262L1
1mg52,00€5mg114,00€10mg172,00€25mg284,00€50mg411,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)138,00€Flesinoxan
CAS:Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Fórmula:C22H26FN3O4Forma y color:SolidPeso molecular:415.46Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Fórmula:C22H23N3O2Pureza:98.06% - 99%Forma y color:SolidPeso molecular:361.44VA012
CAS:VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. It has been shown to reduce food intake and prevent weight gain during subchronic administration without causing central nervous system-related discomfort. VA012 is applicable in obesity research.Fórmula:C21H19N3Forma y color:SolidPeso molecular:313.40
