Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Ro60-0175
CAS:Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.Fórmula:C11H12ClFN2Pureza:97.09%Forma y color:SolidPeso molecular:226.68Ref: TM-T39161
1mg87,00€5mg216,00€10mg354,00€25mg620,00€50mg847,00€100mg1.169,00€1mL*10mM (DMSO)197,00€5-HT3 antagonist 3
CAS:5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).Fórmula:C20H21N3OPureza:99.69%Forma y color:SolidPeso molecular:319.4Ref: TM-T10162
1mg115,00€2mg172,00€5mg255,00€10mg375,00€25mg562,00€50mg792,00€100mg1.064,00€500mgA consultarElzasonan hydrochloride
CAS:Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in the study of depression.Fórmula:C22H24Cl3N3OSForma y color:SolidPeso molecular:484.87ASP-2205
CAS:ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), enhances the urethral closure reflex mediated by the genital nerve, thereby preventing urinary incontinence.Fórmula:C19H28N2OForma y color:SolidPeso molecular:300.44NAN-190 hydrobromide
CAS:NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.Fórmula:C23H28BrN3O3Pureza:95.92%Forma y color:SolidPeso molecular:474.39BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Forma y color:SolidPeso molecular:458.42R 59-022 hydrochloride
CAS:R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.Fórmula:C27H27ClFN3OSPureza:97.7%Forma y color:SolidPeso molecular:496.04Desvenlafaxine
CAS:Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Fórmula:C16H25NO2Pureza:99.46% - 99.81%Forma y color:White Crystalline PowderPeso molecular:263.38Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Fórmula:C23H24FN3O2Pureza:99.20%Forma y color:SolidPeso molecular:393.4525E-NBOMe hydrochloride
CAS:25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.Fórmula:C20H28ClNO3Forma y color:SolidPeso molecular:365.89R-137696
CAS:R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal stomach. It is utilized in research related to functional dyspepsia.Fórmula:C17H23N3O2Forma y color:SolidPeso molecular:301.38AAZ-A 154
CAS:AAZ-A 154 is a selective, competitive, and non-hallucinogenic antagonist of the 5-HT2AR. It promotes neuronal growth in rodents and results in lasting beneficial behavioral effects.Fórmula:C14H20N2OForma y color:SolidPeso molecular:232.32AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.Fórmula:C24H33BrN2O2Pureza:98%Forma y color:SolidPeso molecular:461.44Roluperidone
CAS:Roluperidone (CYR-101) is a novel cyclic amide derivative.Fórmula:C22H23FN2O2Pureza:96.46% - 97.77%Forma y color:SolidPeso molecular:366.43Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Fórmula:C21H33Cl3N4OPureza:100% - 98.52%Forma y color:SolidPeso molecular:463.87Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Forma y color:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Palonosetron hydrochloride
CAS:Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Forma y color:White SolidPeso molecular:332.87Sevoflurane
CAS:Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Fórmula:C4H3F7OPureza:99.78%Forma y color:Less Oil Colorless OilPeso molecular:200.05Ref: TM-T22425
2mg42,00€5mg57,00€10mg80,00€25mg116,00€50mg166,00€100mg240,00€200mg359,00€1mL*10mM (DMSO)59,00€Zalospirone
CAS:Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Fórmula:C24H29N5O2Pureza:100% - 99%Forma y color:SolidPeso molecular:419.52ALEPH hydrochloride
CAS:ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Fórmula:C12H20ClNO2SForma y color:SolidPeso molecular:277.81
