Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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TIK-301
CAS:TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nMFórmula:C14H17ClN2O2Pureza:98%Forma y color:SolidPeso molecular:280.75Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Fórmula:C26H35NO7Pureza:98.53% - 99.43%Forma y color:CoaPeso molecular:473.57Clomipramine
CAS:Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.Fórmula:C19H23ClN2Pureza:99.31%Forma y color:SolidPeso molecular:314.85Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Fórmula:C15H19N5Pureza:99.74%Forma y color:SolidPeso molecular:269.35WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Fórmula:C25H34N4O2·C4H4O4Pureza:99.26% - 99.68%Forma y color:SolidPeso molecular:538.64Ref: TM-T2631
2mg46,00€5mg66,00€10mg95,00€25mg180,00€50mg334,00€100mg495,00€200mg717,00€500mg1.111,00€1mL*10mM (DMSO)79,00€Sertraline hydrochloride
CAS:Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.Fórmula:C17H18Cl3NPureza:99.12% - 99.89%Forma y color:Solid PowderPeso molecular:342.691Ref: TM-T0482
5mg51,00€10mg63,00€25mg103,00€50mg180,00€100mg235,00€200mg304,00€500mg515,00€1mL*10mM (DMSO)57,00€4-Bromo-2,5-DMMA
CAS:4-Bromo-2,5-DMMA (Compound 2) demonstrates affinity for the 5-HT2 binding site and has an ED50 of 0.82 mg/kg in rat discrimination experiments.Fórmula:C12H18BrNO2Forma y color:SolidPeso molecular:288.18SB 699551 dihydrochloride
CAS:SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Fórmula:C34H47Cl2N3OPureza:96.53%Forma y color:SolidPeso molecular:584.66Ref: TM-T23325
1mg52,00€5mg111,00€10mg180,00€25mg311,00€50mg449,00€100mg615,00€1mL*10mM (DMSO)150,00€Tianeptine sodium salt
CAS:Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H24ClN2NaO4SPureza:99.82%Forma y color:SolidPeso molecular:458.93Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Fórmula:C18H22N2SPureza:99.34% - 99.34%Forma y color:SolidPeso molecular:298.45Ref: TM-T2395
1g505,00€10mg50,00€25mg69,00€50mg95,00€100mg124,00€200mg215,00€500mg350,00€1mL*10mM (DMSO)48,00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Fórmula:C23H30N4O2SPureza:99.23%Forma y color:White PowderPeso molecular:426.57Tropisetron hydrochloride
CAS:Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.Fórmula:C17H21ClN2O2Pureza:99.72% - 99.83%Forma y color:SolidPeso molecular:320.82Cinanserin hydrochloride
CAS:Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.Fórmula:C20H25ClN2OSPureza:99.32%Forma y color:SolidPeso molecular:376.94Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Fórmula:C20H20ClF5N2OPureza:99.97%Forma y color:SolidPeso molecular:434.83Ref: TM-T22936
1mg64,00€2mg87,00€5mg116,00€10mg167,00€25mg283,00€50mg424,00€100mg598,00€200mg805,00€1mL*10mM (DMSO)125,00€3-AQC
CAS:3-AQC is a competitive antagonist of 5-HT3.Fórmula:C20H21N5O4Pureza:99.45%Forma y color:SolidPeso molecular:395.41Ref: TM-T8475
2mg35,00€5mg50,00€10mg66,00€25mg95,00€50mg140,00€100mg205,00€200mg304,00€1mL*10mM (DMSO)57,00€Rodatristat ethyl
CAS:Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.Fórmula:C29H31ClF3N5O3Pureza:98%Forma y color:SolidPeso molecular:590.04LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Fórmula:C21H25ClN2O2Pureza:99.47%Forma y color:SolidPeso molecular:372.89Seganserin
CAS:Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.Fórmula:C29H27F2N3OPureza:98%Forma y color:SolidPeso molecular:471.54PRX-08066
CAS:PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Fórmula:C19H17ClFN5SPureza:98.04% - 98.07%Forma y color:SolidPeso molecular:401.89Ref: TM-T16669
1mg60,00€5mg119,00€10mg170,00€25mg350,00€50mg522,00€100mg748,00€200mg1.026,00€1mL*10mM (DMSO)111,00€Vabicaserin hydrochloride
CAS:Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).Fórmula:C15H21ClN2Pureza:98.32%Forma y color:SolidPeso molecular:264.79Ref: TM-T13275
1mg84,00€5mg178,00€10mg264,00€25mg424,00€50mg562,00€100mg775,00€200mg1.026,00€1mL*10mM (DMSO)188,00€
