Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Fórmula:C20H33NO7Pureza:99.26%Forma y color:White Crystalline PowdePeso molecular:399.48Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Forma y color:SolidPeso molecular:438.49cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44Ebalzotan
CAS:NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.Fórmula:C19H30N2O2Pureza:99.08% - 99.41%Forma y color:SolidPeso molecular:318.45Relenopride
CAS:YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to study irritable bowel syndrome with constipation.Fórmula:C24H30ClFN4O4Pureza:98.91% - 99.20%Forma y color:SoildPeso molecular:492.97MM 77 dihydrochloride
CAS:MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.Fórmula:C19H29Cl2N3O3Pureza:100.00%Forma y color:SolidPeso molecular:418.36Ref: TM-T23007
1mg86,00€5mg157,00€10mg215,00€25mg472,00€50mg687,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)281,00€AL 34662
CAS:AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFórmula:C10H13N3OPureza:99.77%Forma y color:SolidPeso molecular:191.23Naluzotan hydrochloride
CAS:Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.Fórmula:C23H39ClN4O3SPureza:98.61%Forma y color:SolidPeso molecular:487.1PNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFórmula:C13H17ClN2Pureza:97.83%Forma y color:SolidPeso molecular:236.74RS-67333
CAS:RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Fórmula:C19H29ClN2O2Pureza:99.24%Forma y color:SolidPeso molecular:352.9(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Fórmula:C12H14O5Pureza:99.83%Forma y color:SolidPeso molecular:238.24Clovoxamine
CAS:Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.Fórmula:C14H21ClN2O2Pureza:98.88% - 99.16%Forma y color:SolidPeso molecular:284.78Mosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFórmula:C21H25ClFN3O3Pureza:99.56%Forma y color:White To Off-White Crystalline SolidPeso molecular:421.89SB 216641 hydrochloride
CAS:SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.Fórmula:C28H31ClN4O4Pureza:98.40% - 99.23%Forma y color:SolidPeso molecular:523.02Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:99.94%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Fórmula:C26H27N5O2Pureza:99.61%Forma y color:Light Yellow SolidPeso molecular:441.52Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, andFórmula:C19H23NO8Forma y color:SolidPeso molecular:393.39LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Fórmula:C30H34N4OPureza:98.65%Forma y color:SolidPeso molecular:466.62Ref: TM-T5387
2mg47,00€5mg70,00€10mg96,00€25mg180,00€50mg305,00€100mg487,00€200mg695,00€1mL*10mM (DMSO)77,00€Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Forma y color:SolidPeso molecular:383.49Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Fórmula:C20H25NOPureza:99.52%Forma y color:SolidPeso molecular:295.42Ref: TM-T22964
1mg40,00€5mg88,00€10mg126,00€25mg273,00€50mg432,00€100mg638,00€500mg1.359,00€1mL*10mM (DMSO)88,00€
