Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Fórmula:C19H28Cl2N6O2Pureza:99% - 99.89%Forma y color:SolidPeso molecular:443.37Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Fórmula:C16H19NOPureza:99.12%Forma y color:SolidPeso molecular:241.33Ref: TM-T67956
1mg97,00€5mg217,00€10mg325,00€25mg557,00€50mg797,00€100mg1.103,00€500mg2.205,00€1mL*10mM (DMSO)188,00€RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Fórmula:C20H25ClN2O2Pureza:98%Forma y color:SolidPeso molecular:360.88VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Fórmula:C13H15ClN4Pureza:99.66%Forma y color:SolidPeso molecular:262.74Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Fórmula:C19H23Cl2N5OPureza:99.50% - 99.52%Forma y color:SolidPeso molecular:408.335-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stabilityFórmula:C17H22F2N6OPureza:98%Forma y color:SolidPeso molecular:364.39Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Ref: TM-T4577
1mg51,00€5mg108,00€10mg180,00€25mg316,00€50mg472,00€100mg658,00€200mg938,00€1mL*10mM (DMSO)108,00€Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Fórmula:C15H23NOPureza:99.11% - 99.13%Forma y color:SolidPeso molecular:233.35Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Fórmula:C19H21N3SPureza:97.01%Forma y color:SolidPeso molecular:323.46Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Forma y color:SolidPeso molecular:449.4p-MPPF dihydrochloride
CAS:p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.Fórmula:C25H29Cl2FN4O2Pureza:99.78%Forma y color:SolidPeso molecular:507.43Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Fórmula:C20H21FN2OPureza:99.89%Forma y color:SolidPeso molecular:324.39AGH-107
CAS:AGH-107 is a highly selective 5-HT7 receptor agonist that can cross the blood-brain barrier, featuring a Ki value of 6 nM and an EC50 value of 19 nM. Demonstrating high selectivity for central nervous system targets, AGH-107 also exhibits high metabolic stability and low toxicity in HEK-293 and HepG2 cell cultures.Fórmula:C13H12IN3Forma y color:SolidPeso molecular:337.162-Methyl-5-HT
CAS:2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Fórmula:C11H14N2OPureza:95.64%Forma y color:SolidPeso molecular:190.24Ref: TM-T10075
5mg50,00€10mg88,00€25mg187,00€50mg354,00€100mg528,00€500mg1.159,00€1mL*10mM (DMSO)52,00€Pumosetrag Hydrochloride
CAS:Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.Fórmula:C15H18ClN3O2SPureza:98%Forma y color:SolidPeso molecular:339.845HT6-ligand-1
CAS:5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Fórmula:C20H22BrN3O2SPureza:98.48% - 98.95%Forma y color:SolidPeso molecular:448.38Remlifanserin
CAS:Remlifanserin is a potent inverse agonist of the serotonin receptor (5-HT2A).Fórmula:C24H29F2N3O2Forma y color:SolidPeso molecular:429.50S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Fórmula:C24H27ClFN3O2Pureza:99.5%Forma y color:SolidPeso molecular:443.945-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Fórmula:C18H21N3OPureza:98%Forma y color:SolidPeso molecular:295.38Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Fórmula:C24H25FN4O2Pureza:99.33%Forma y color:SolidPeso molecular:420.48
