AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Formula:C19H32N2O2·2HClPurity:98%Color and Shape:SolidMolecular weight:393.4Ethyl (triphenylphosphoranylidene) acetate
CAS:Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.Formula:C22H21O2PPurity:98.43%Color and Shape:White Or Slight Yellow PowderMolecular weight:348.37YM-58790
CAS:YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.Formula:C27H31N3O2Purity:99%Color and Shape:SoildMolecular weight:429.55Oxotremorine sesquifumarate
CAS:Oxotremorine sesquifumarate is a muscarinic agonist.Formula:C12H18N2OC4H4O4Purity:99.94%Color and Shape:SolidMolecular weight:380.395-AAM-2-CP
CAS:5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.Formula:C8H9ClN2OPurity:98.62%Color and Shape:SolidMolecular weight:184.62Piperidolate
CAS:Piperidolate inhibits intestinal cramp induced by acetylcholineFormula:C21H25NO2Purity:98.45%Color and Shape:SolidMolecular weight:323.43Varenicline dihydrochloride
CAS:Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.Formula:C13H15Cl2N3Purity:99.21%Color and Shape:SolidMolecular weight:284.18GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurity:98.76%Color and Shape:SolidMolecular weight:405.31Desfesoterodine
CAS:Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.Formula:C22H31NO2Purity:100%Color and Shape:SolidMolecular weight:341.49Ref: TM-T6364
1mg66.00€5mg144.00€10mg216.00€25mg373.00€50mg550.00€100mg792.00€500mg1,605.00€1mL*10mM (DMSO)159.00€Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purity:98%Color and Shape:SolidMolecular weight:538.6(S)-Coclaurine
CAS:(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.Formula:C17H19NO3Purity:97.72%Color and Shape:SolidMolecular weight:285.34Rivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.Formula:C10H16Cl2N2Purity:99.76%Color and Shape:SoildMolecular weight:235.15Ref: TM-T12738L1
1mg35.00€5mg74.00€10mg105.00€25mg246.00€50mg444.00€100mg650.00€1mL*10mM (DMSO)116.00€Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Formula:C23H26N2O2·C4H6O4Purity:99.85% - 99.98%Color and Shape:SolidMolecular weight:480.56TC-T 6000
CAS:TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.Formula:C26H48N8O2Purity:98.14%Color and Shape:SolidMolecular weight:504.71Tolterodine tartrate
CAS:Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.Formula:C22H31NO·C4H6O6Purity:99.95%Color and Shape:White-To-Off-White Crystalline PowderMolecular weight:475.58Thiacloprid
CAS:Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.Formula:C10H9ClN4SPurity:98.66%Color and Shape:Yellowish Crystalline PowderMolecular weight:252.72Fesoterodine
CAS:Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.Formula:C26H37NO3Purity:96.27% - 97.1%Color and Shape:SolidMolecular weight:411.58CB-7921220
CAS:CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.Formula:C14H12N2O2Purity:99.57%Color and Shape:SolidMolecular weight:240.26(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Formula:C24H17ClF2N2O2Purity:98.83%Color and Shape:SolidMolecular weight:438.85mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formula:C23H26ClIN2O2Purity:99.87%Color and Shape:SolidMolecular weight:524.82Ref: TM-T5655
1mg52.00€5mg116.00€10mg183.00€25mg324.00€50mg449.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)135.00€
