AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Carbaryl
CAS:Carbaryl is a carbamate insecticide/parasiticide with low dermal toxicity used against head lice.Formula:C12H11NO2Purity:98.26% - 99.75%Color and Shape:Colorless To Light Tan Crystals By Inhalation (Dust Etc ) Produces Toxic Oxides Of Nitrogen During CombustionMolecular weight:201.22Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurity:99.20%Color and Shape:SolidMolecular weight:320.84Ref: TM-T7193
1mg73.00€5mg140.00€10mg220.00€25mg369.00€50mg523.00€100mg712.00€200mg938.00€1mL*10mM (DMSO)153.00€(±)-Acetylcarnitine chloride
CAS:(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.Formula:C9H18ClNO4Purity:99.98%Color and Shape:White Crystalline PowderMolecular weight:239.7Tiquizium
CAS:Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.Formula:C19H24NS2Purity:99.02%Color and Shape:SolidMolecular weight:330.53Ref: TM-T9877
1mg77.00€5mg155.00€10mg220.00€25mg338.00€50mg472.00€100mg632.00€200mg853.00€1mL*10mM (DMSO)157.00€SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Formula:C25H31N3O2SPurity:98.3% - 99.62%Color and Shape:SolidMolecular weight:437.6S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurity:99.72%Color and Shape:SolidMolecular weight:418.07Ref: TM-T23286
5mg47.00€10mg70.00€25mg145.00€50mg226.00€100mg356.00€200mg507.00€1mL*10mM (DMSO)50.00€UB 165 fumarate
CAS:UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.Formula:C17H19ClN2O4Purity:98.91%Color and Shape:SolidMolecular weight:350.8AQW051
CAS:AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formula:C19H22N2OPurity:99.67%Color and Shape:SolidMolecular weight:294.39Ref: TM-T26646
1mg35.00€2mg48.00€5mg70.00€10mg104.00€25mg216.00€50mg329.00€100mg464.00€500mg1,008.00€1mL*10mM (DMSO)71.00€Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purity:98.12%Color and Shape:SolidMolecular weight:597.75Neostigmine methyl sulfate
CAS:Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.Formula:C13H22N2O6SPurity:99.34% - 99.53%Color and Shape:Crystalline SolidMolecular weight:334.39Simpinicline
CAS:Simpinicline (OC-02) (OC-02) is an nAChR agonist that activates the trigeminal parasympathetic pathway and can be used to treat dry eye.Formula:C10H13N3Purity:98.54% - 99.63%Color and Shape:SolidMolecular weight:175.23SSR 180
CAS:SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.Formula:C14H17BrN2O2Purity:98.95%Color and Shape:SoildMolecular weight:325.20Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Formula:C65H82N2O18S2Purity:98% - 99.71%Color and Shape:SolidMolecular weight:1243.49Ref: TM-T6397
10mg35.00€25mg52.00€50mg66.00€100mg100.00€200mg155.00€500mg240.00€1mL*10mM (DMSO)55.00€Terodiline
CAS:Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.Formula:C20H27NPurity:98.50% - 99.41%Color and Shape:SolidMolecular weight:281.44Isopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.Formula:C23H33IN2OPurity:99.91%Color and Shape:SolidMolecular weight:480.43Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formula:C18H27ClN2O4Purity:98.94%Color and Shape:SolidMolecular weight:370.87Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFormula:C9H15NO2Purity:100%Color and Shape:SolidMolecular weight:169.22Phenserine
CAS:Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.Formula:C20H23N3O2Purity:98%Color and Shape:SolidMolecular weight:337.42NS3861
CAS:NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Formula:C12H14BrNSPurity:99.40%Color and Shape:SolidMolecular weight:284.22Dicyclomine hydrochloride
CAS:Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.Formula:C19H36ClNO2Purity:99.81%Color and Shape:SolidMolecular weight:345.95
