AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Fesoterodine fumarate
CAS:Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.Formula:C26H37NO3·C4H4O4Purity:98% - 98.55%Color and Shape:White SolidMolecular weight:527.65Blarcamesine
CAS:Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.Formula:C19H23NOPurity:99.87%Color and Shape:SolidMolecular weight:281.39Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H17ClN2OS·HClPurity:98.34% - 99.85%Color and Shape:SolidMolecular weight:357.3PQCA
CAS:PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.Formula:C22H20N4O3Purity:98.95%Color and Shape:SolidMolecular weight:388.42(-)-Coclaurine hydrochloride
CAS:(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.Formula:C17H20ClNO3Purity:97.75%Color and Shape:SoildMolecular weight:321.8Ref: TM-TN1519L
1mg115.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€1mL*10mM (DMSO)249.00€Temephos
CAS:Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.Formula:C16H20O6P2S3Purity:≥95%Color and Shape:White Crystalline Solid Or LiquidMolecular weight:466.47ASM-024
CAS:ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Formula:C15H25N2Purity:99.79%Color and Shape:SolidMolecular weight:233.37Ref: TM-T26666
1mg245.00€5mg610.00€10mg868.00€25mg1,301.00€50mg1,758.00€100mg2,375.00€500mg4,655.00€1mL*10mM (DMSO)507.00€Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Formula:C7H17N2O2·ClPurity:95% - 99.73%Color and Shape:White CrystallineMolecular weight:196.68PSEM 89S TFA
CAS:PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.Formula:C18H23F3N2O5Purity:99.90%Color and Shape:SolidMolecular weight:404.38Meseclazone
CAS:Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.Formula:C11H10ClNO3Purity:98%Color and Shape:SolidMolecular weight:239.65Rocuronium bromide
CAS:Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.Formula:C32H53BrN2O4Purity:100% - 99.77%Color and Shape:White Or Off-White PowderMolecular weight:609.68NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formula:C14H9Cl2F3N2O2Purity:99.11%Color and Shape:SolidMolecular weight:365.13VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purity:97.56%Color and Shape:SolidMolecular weight:316.15Asoxime dichloride
CAS:Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.Formula:C14H16Cl2N4O3Purity:99.86%Color and Shape:SolidMolecular weight:359.21Timepidium bromide
CAS:Timepidium bromide is an agent of anticholinergic.Formula:C17H22BrNOS2Purity:98%Color and Shape:SolidMolecular weight:400.4PHA 568487 free base
CAS:PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.Formula:C16H20N2O3Purity:99.74%Color and Shape:SolidMolecular weight:288.34OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.49%Color and Shape:SolidMolecular weight:330.44Posatirelin
CAS:Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.Formula:C17H28N4O4Purity:97.41% - 98.22%Color and Shape:SolidMolecular weight:352.43CDD0102
CAS:CDD0102 is a potent agonist of M1 Muscarinic receptor.Formula:C8H12N4OPurity:98%Color and Shape:SolidMolecular weight:180.21Decamethonium bromide
CAS:Decamethonium bromide (Syncurine) is a neuromuscular blocker and nicotinic AChR partial agonist.Formula:C16H38Br2N2Purity:99.90%Color and Shape:Physical Description Crystals Derived From Methanol And Acetone (Ntp 1992)Molecular weight:418.29
