AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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hBChE-IN-2
CAS:hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.Formula:C27H36N4O3Purity:99.69% - 99.86%Color and Shape:SoildMolecular weight:464.6(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purity:97.4%Color and Shape:SolidMolecular weight:236.142Ref: TM-T12653
1mg52.00€2mg74.00€5mg96.00€10mg169.00€25mg323.00€50mg497.00€100mg720.00€1mL*10mM (DMSO)119.00€3-Bromocytisine
CAS:3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).Formula:C11H13BrN2OPurity:98.14%Color and Shape:SolidMolecular weight:269.14Ref: TM-T10108
1mg95.00€5mg227.00€10mg309.00€25mg520.00€50mg748.00€100mg1,026.00€1mL*10mM (DMSO)208.00€W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formula:C32H44Br2N4O4Purity:95.56%Color and Shape:SolidMolecular weight:708.52Cyclodrine
CAS:Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.Formula:C19H29NO3Purity:98.3%Color and Shape:SoildMolecular weight:319.44Ref: TM-T10914L
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)157.00€S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purity:98.43%Color and Shape:SolidMolecular weight:674.01VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formula:C18H28ClN3O3Purity:99% - 99.97%Color and Shape:SolidMolecular weight:369.89BuChE-IN-TM-10
CAS:TM-10: Potent BuChE inhibitor, IC50 8.9 nM, disaggregates Aβ, antioxidant, BBB penetrant, may treat Alzheimer's.Formula:C32H38N2O3Purity:99.16%Color and Shape:SolidMolecular weight:498.66Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purity:99.89%Color and Shape:White Crystalline PowderMolecular weight:202.21CDD0102 HCl
CAS:CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.Formula:C8H13ClN4OPurity:99.7%Color and Shape:SoildMolecular weight:216.67Desformylflustrabromine hydrochloride
CAS:Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.Formula:C17H12INO5Purity:98.51%Color and Shape:SolidMolecular weight:437.19Ipratropium bromide monohydrate
CAS:Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.Formula:C20H32BrNO4Purity:97.85%Color and Shape:SolidMolecular weight:430.38SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formula:C14H18BrClN2O2Purity:99.77%Color and Shape:SolidMolecular weight:361.669-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purity:99.85%Color and Shape:SolidMolecular weight:203.24ICL-CCIC-0019
CAS:ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.Formula:C26H44Br2N4Purity:97.62%Color and Shape:SolidMolecular weight:572.46Ref: TM-T27579
1mg185.00€5mg415.00€10mg613.00€25mg938.00€50mg1,311.00€100mg1,768.00€500mg3,535.00€1mL*10mM (DMSO)545.00€VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Formula:C18H19N3O2SPurity:99.56%Color and Shape:SolidMolecular weight:341.43Ref: TM-T17238
1mg40.00€5mg88.00€10mg118.00€25mg254.00€50mg406.00€100mg612.00€200mg842.00€1mL*10mM (DMSO)99.00€Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurity:99.84%Color and Shape:White Crystalline PowderMolecular weight:322.83Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:100% - 99.76%Color and Shape:White SolidMolecular weight:203.75Isoxazole
CAS:Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and inhibit the Sxc- antiporter.Formula:C3H3NOPurity:99.34%Color and Shape:Colorless LiquidMolecular weight:69.06Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C25H26F4N2O8Purity:99.86%Color and Shape:SolidMolecular weight:558.48
