AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Formula:C21H21N3O2Purity:99.9%Color and Shape:SolidMolecular weight:347.41Ref: TM-T10961
1mg215.00€5mg426.00€10mg598.00€25mg889.00€50mg1,188.00€100mg1,605.00€1mL*10mM (DMSO)472.00€Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Formula:C24H26ClNO4Purity:99.78%Color and Shape:White SolidMolecular weight:427.92Rivastigmine tartrate
CAS:Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.Formula:C14H22N2O2·C4H6O6Purity:98% - 99.66%Color and Shape:White To Off-White PowderMolecular weight:400.43Methyllycaconitine citrate
CAS:Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.Formula:C43H58N2O17Purity:98.03% - 98.91%Color and Shape:SolidMolecular weight:874.92Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Formula:C21H28BrNO3Purity:99.29%Color and Shape:SolidMolecular weight:422.36Homatropine Methylbromide
CAS:Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.Formula:C17H24BrNO3Purity:98.97%Color and Shape:SolidMolecular weight:370.299-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.41%Color and Shape:SolidMolecular weight:163.18Trihexyphenidyl hydrochloride
CAS:Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.Formula:C20H32ClNOPurity:99.65%Color and Shape:SolidMolecular weight:337.927Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purity:98.88%Color and Shape:SolidMolecular weight:362.83Ref: TM-T9771
1mg66.00€5mg145.00€10mg226.00€25mg408.00€50mg558.00€100mg787.00€200mg1,035.00€1mL*10mM (DMSO)160.00€Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Formula:C14H23N3OSPurity:99.61%Color and Shape:SolidMolecular weight:281.42Ref: TM-T36640
2mg38.00€5mg55.00€10mg93.00€25mg165.00€50mg264.00€100mg420.00€200mg607.00€1mL*10mM (DMSO)60.00€Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formula:C28H30N2O2Purity:99.78%Color and Shape:SolidMolecular weight:426.55BQCA
CAS:BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.Formula:C18H15NO4Purity:97.22%Color and Shape:SolidMolecular weight:309.32Tematropium
CAS:Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.Formula:C21H31NO8SPurity:98.87%Color and Shape:SolidMolecular weight:457.54Ref: TM-T10732
1mg212.00€2mg284.00€5mg449.00€10mg615.00€25mg929.00€50mg1,244.00€100mg1,691.00€1mL*10mM (DMSO)507.00€Tiotropium bromide
CAS:Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).Formula:C19H22BrNO4S2Purity:96.82% - 99.63%Color and Shape:White SolidMolecular weight:472.42Propoxur
CAS:Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.Formula:C11H15NO3Purity:98.15% - 99.87%Color and Shape:Minute Crystals (Niosh 2016)Molecular weight:209.24Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formula:C22H32BrNO5Purity:98.85%Color and Shape:SolidMolecular weight:470.4Ref: TM-T28827
1mg74.00€5mg160.00€10mg250.00€25mg452.00€50mg680.00€100mg1,008.00€200mg1,349.00€1mL*10mM (DMSO)170.00€Tribendimidine
CAS:Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.Formula:C28H32N6Purity:≥98%Color and Shape:SolidMolecular weight:452.59Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Formula:C29H34BrNO2Purity:98.40% - 99.09%Color and Shape:SolidMolecular weight:508.49Ref: TM-T4997
1mg40.00€2mg52.00€5mg85.00€10mg124.00€25mg212.00€50mg350.00€100mg525.00€1mL*10mM (DMSO)87.00€VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Formula:C17H12F3NO4Purity:100%Color and Shape:SolidMolecular weight:351.28Ref: TM-T8007
2mg35.00€5mg52.00€10mg86.00€25mg144.00€50mg227.00€100mg359.00€500mg838.00€1mL*10mM (DMSO)58.00€
