AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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bPiDDB
CAS:bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.Formula:C24H38Br2N2Purity:98.72%Color and Shape:SolidMolecular weight:514.38Ref: TM-T37818
2mg43.00€5mg60.00€10mg96.00€25mg188.00€50mg278.00€100mg411.00€200mg607.00€1mL*10mM (DMSO)73.00€Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Formula:C24H40O10S2Purity:98%Color and Shape:SolidMolecular weight:552.7Loxeen
CAS:Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.Formula:C20H25NO·CH4O3SPurity:99.46%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.52Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Formula:C24H31N5O2Purity:99.81%Color and Shape:SolidMolecular weight:421.54Cimetropium Bromide
CAS:Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.Formula:C21H28BrNO4Color and Shape:SolidMolecular weight:438.36Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formula:C17H17N5O6SPurity:98.83% - 99.69%Color and Shape:Off-White SolidMolecular weight:419.414-DAMP
CAS:4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.Formula:C21H26INO2Purity:98%Color and Shape:SolidMolecular weight:451.34Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Formula:C20H21N3OPurity:99.17%Color and Shape:SolidMolecular weight:319.4Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Formula:C22H31NOPurity:99.71%Color and Shape:White Like Or Light Brown Crystalline PowderMolecular weight:325.49Mepenzolate Bromide
CAS:Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.Formula:C21H26BrNO3Purity:95.73% - 99.21%Color and Shape:SolidMolecular weight:420.34Aclidinium bromide
CAS:Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.Formula:C26H30NO4S2·BrPurity:98.93% - 99.69%Color and Shape:SolidMolecular weight:564.55Ref: TM-T2555
2mg39.00€5mg57.00€10mg88.00€25mg145.00€50mg234.00€100mg350.00€500mg825.00€1mL*10mM (DMSO)72.00€Clidinium bromide
CAS:Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.Formula:C22H26BrNO3Purity:98.89% - 99.86%Color and Shape:White Crystalline SolidMolecular weight:432.35SQ22536
CAS:SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.Formula:C9H11N5OPurity:99.18%Color and Shape:Off-White SolidMolecular weight:205.22SCH-900271
CAS:SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.Formula:C14H16N2O4Purity:98.25% - 99%Color and Shape:SolidMolecular weight:276.29Ref: TM-T34573
1mg118.00€5mg275.00€10mg419.00€25mg692.00€50mg938.00€100mg1,320.00€500mg2,632.00€1mL*10mM (DMSO)263.00€Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Formula:C23H27ClN2O2Purity:99.32%Color and Shape:Off-White PowderMolecular weight:398.93Oxitropium Bromide
CAS:Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.Formula:C19H26BrNO4Purity:98%Color and Shape:SolidMolecular weight:412.32Nanofin
CAS:Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.Formula:C7H15NPurity:99.818%Color and Shape:Clear Colorless To Slightly Yellow LiquidMolecular weight:113.2AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Formula:C27H38N6O2Purity:98%Color and Shape:SolidMolecular weight:478.63TAK-071
CAS:TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).Formula:C24H24FN3O3Purity:98.02%Color and Shape:SolidMolecular weight:421.46Carbachol
CAS:Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.Formula:C6H15ClN2O2Purity:100% - 90%Color and Shape:SolidMolecular weight:182.65
