AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Products of "AChR"
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Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purity:99.87%Color and Shape:SolidMolecular weight:362.46Vecuronium bromide
CAS:Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscleFormula:C34H57BrN2O4Purity:99.63% - 99.92%Color and Shape:White PowderMolecular weight:637.73VU0453595
CAS:VU0453595 is a M1 positive allosteric modulator (PAM).Formula:C18H15FN4OPurity:99.48%Color and Shape:SolidMolecular weight:322.34Lupinine
CAS:Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.Formula:C10H19NOPurity:99.95%Color and Shape:SolidMolecular weight:169.26Ref: TM-FR16605
1mg95.00€5mg180.00€10mg271.00€25mg462.00€50mg672.00€100mg918.00€500mg1,840.00€1ml*10 (DMSO)151.00€Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formula:C10H21NPurity:98.18% - 99.92%Color and Shape:Colorless - Light Yellow Clear LiquidMolecular weight:155.28Atropine methyl bromide
CAS:Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.Formula:C18H26BrNO3Purity:99.70%Color and Shape:SolidMolecular weight:384.308Ref: TM-T14345
1mg35.00€5mg70.00€10mg105.00€25mg187.00€50mg274.00€100mg404.00€200mg587.00€1mL*10mM (DMSO)77.00€Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formula:C16H20N2O2Purity:98.63%Color and Shape:SolidMolecular weight:272.34Ref: TM-T22380
1mg93.00€2mg126.00€5mg187.00€10mg283.00€25mg462.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)187.00€Zamifenacin fumarate
CAS:Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.Formula:C31H33NO7Purity:99.78%Color and Shape:SolidMolecular weight:531.6Ref: TM-T13385
1mg40.00€5mg88.00€10mg119.00€25mg216.00€50mg354.00€100mg533.00€200mg743.00€1mL*10mM (DMSO)93.00€RPR121056
CAS:RPR121056 is a Irinotecan metabolite, which is generated by CYP3A4. Irinotecan is an antineoplastic agent that inhibits topoisomerase type I.Formula:C33H38N4O8Purity:98%Color and Shape:SolidMolecular weight:618.68GSK-1034702
CAS:GSK-1034702 is an M1 mAChR agonist that improves cognitive deficits and may be useful in the study of neurologic disorders.Formula:C18H24FN3O2Purity:99.69%Color and Shape:SolidMolecular weight:333.4Sch412348
CAS:Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.Formula:C22H21F2N9OPurity:98%Color and Shape:SolidMolecular weight:465.46Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Formula:C9H12Cl2N2OPurity:95% - 98.71%Color and Shape:SolidMolecular weight:235.11(Rac)-Sabcomeline
CAS:(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.Formula:C10H15N3OPurity:99.14%Color and Shape:SolidMolecular weight:193.25Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purity:99.46%Color and Shape:White To Off-White SolidMolecular weight:525.59VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurity:98.46%Color and Shape:SolidMolecular weight:355.41GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purity:98%Color and Shape:SolidMolecular weight:308.37TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.Formula:C25H32N4OPurity:97.87% - 99.9%Color and Shape:SolidMolecular weight:404.55NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Formula:C27H44ClNO8Purity:98% - 98%Color and Shape:SolidMolecular weight:546.09TZ3O
CAS:TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type model in rats.Formula:C18H13NO4SPurity:99.84%Color and Shape:SolidMolecular weight:339.37Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Formula:C21H26ClNO2Purity:99.50%Color and Shape:SolidMolecular weight:359.89
